SCHEMBL7914828

SCHEMBL7914828

COc1cc(C(=O)NC(C)(C)C)ccc1S(=O)(=O)n1nc(C2CC2)n(C2CC2)c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 1/20 0.39
ALDH1A1 P00352 2/20 0.38
KMT2A Q03164 3/20 0.37
LRRK2 Q5S007 1/20 0.35
HPGD P15428 1/20 0.35
LMNA P02545 3/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
RAB9A P51151 2/20 0.34
AKR1C3 P42330 2/20 0.34
MEN1 O00255 2/20 0.34
MAPT P10636 2/20 0.34
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
HSD11B1 P28845 1/20 0.34
TP53 P04637 1/20 0.34
PTK2 Q05397 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7911467 0.89 ALDH1A1 (0.39) AVPR1AALDH1A1KMT2ALRRK2HPGD
SCHEMBL16167675 0.89 ALDH1A1 (0.39) AVPR1AALDH1A1KMT2ALRRK2HPGD
SCHEMBL7908197 0.88 ALDH1A1 (0.38) AVPR1AALDH1A1KMT2ALRRK2HPGD
SCHEMBL7908194 0.86 KMT2A (0.38) AVPR1AALDH1A1KMT2ALRRK2HPGD
SCHEMBL7909318 0.86 AVPR1A (0.37) AVPR1AALDH1A1KMT2ALRRK2HPGD
SCHEMBL16167674 0.85 AVPR1A (0.37) AVPR1AALDH1A1KMT2ALRRK2HPGD
SCHEMBL7909327 0.84 AVPR1A (0.39) AVPR1AALDH1A1KMT2ALRRK2HPGD
SCHEMBL16167673 0.84 HSD11B1 (0.40) AVPR1AALDH1A1KMT2ASMN1; SMN2HSD11B1
SCHEMBL7904485 0.78 ALDH1A1 (0.38) AVPR1AALDH1A1KMT2ALMNAMEN1
SCHEMBL7918146 0.77 L3MBTL1 (0.38) AVPR1AALDH1A1KMT2ALRRK2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2373632-B1 SUBSTITUTED BENZYL AND PHENYLSULFONYL TRIAZOLONES, AND USE THEREOF BAYER IP GMBH (DE) 2015-03-04 EP disclosed
US-8859601-B2 Substituted benzyl and phenylsulfonyl triazolones, and use thereof BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-10-14 US disclosed
US-8859601-B2 Substituted benzyl and phenylsulfonyl triazolones, and use thereof BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-10-14 US disclosed
WO-2010063402-A1 SUBSTITUTED BENZYL AND PHENYLSULFONYL TRIAZOLONES, AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-06-10 WO disclosed