SCHEMBL16167698

SCHEMBL16167698

COc1ccc2c(c1)C(CC(=O)O)CC2C

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 8/20 0.49
ATM Q13315 1/20 0.48
FFAR1 O14842 3/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.43
PPARA Q07869 1/20 0.41
LMNA P02545 1/20 0.41
MTNR1A P48039 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PTGS1 P23219 1/20 0.40
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40
FFAR4 Q5NUL3 1/20 0.39
PPARG P37231 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16167706 0.87 MTNR1A (0.42) MTNR1A
SCHEMBL1206528 0.84 PPARD (0.48) PPARDATMFFAR1PTGDR2PPARA
Hydrochloric Acid SCHEMBL1207635 0.83 PPARD (0.47) PPARDATMFFAR1PTGDR2PPARA
SCHEMBL4260242 0.79 MTNR1A (0.65) MTNR1A
Hydrochloric Acid SCHEMBL1396530 0.78 PPARD (0.43) PPARDATMFFAR1PTGDR2PPARA
SCHEMBL31326550 0.77 TP53 (0.41) PPARDATMFFAR1PPARG
SCHEMBL21978182 0.77 TP53 (0.41) PPARDATMFFAR1PPARG
SCHEMBL4264345 0.77 MTNR1A (0.66) MTNR1A
SCHEMBL13891904 0.77 HTR2A (0.40) MTNR1A
SCHEMBL9467265 0.77 MTNR1A (0.52) PPARDMTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8859580-B2 Aryl- and heteroarylcarbonyl derivatives of benzomorphanes and related scaffolds, medicaments containing such compounds and their use BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-10-14 US disclosed