SCHEMBL16197861

SCHEMBL16197861

CN(C(=O)COc1ccc(-n2ccnc2)cc1)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 7/20 0.66
CYP3A4 P08684 5/20 0.66
PORCN Q9H237 4/20 0.66
PDE10A Q9Y233 1/20 0.55
MEN1 O00255 1/20 0.53
ALOX15 P16050 1/20 0.53
TSHR P16473 1/20 0.53
KMT2A Q03164 1/20 0.53
CYP1A2 P05177 6/20 0.50
CYP2C9 P11712 6/20 0.50
CYP2C19 P33261 5/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
LMNA P02545 3/20 0.48
MAPT P10636 2/20 0.48
ALDH1A1 P00352 1/20 0.48
HTT P42858 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
ADH5 P11766 1/20 0.48
CYP19A1 P11511 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16197934 0.79 PORCN (1.00) CYP2D6CYP3A4PORCNMEN1ALOX15
SCHEMBL16201504 0.78 NPC1 (0.59) CYP3A4MEN1KMT2ACYP1A2CYP2C9
SCHEMBL5647696 0.76 RAB9A (0.54) CYP2D6CYP3A4PORCNPDE10AMEN1
SCHEMBL16201462 0.75 PORCN (0.79) CYP2D6CYP3A4PORCNMEN1ALOX15
SCHEMBL5648868 0.75 PDE10A (0.55) CYP2D6CYP3A4PORCNPDE10AMEN1
SCHEMBL16197793 0.75 PORCN (0.74) CYP2D6CYP3A4PORCNMEN1ALOX15
SCHEMBL16201303 0.74 PORCN (0.78) CYP2D6CYP3A4PORCNMEN1ALOX15
SCHEMBL16198312 0.74 PORCN (0.84) CYP2D6CYP3A4PORCNTSHRKMT2A
Ether SCHEMBL6337288 0.74 MEN1 (0.76) CYP2D6CYP3A4PORCNMEN1ALOX15
SCHEMBL5649047 0.73 CYP2D6 (0.52) CYP2D6CYP3A4PORCNPDE10AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014175832-A1 WNT PATHWAY MODULATORS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2014-10-30 WO disclosed
WO-2014175832-A1 WNT PATHWAY MODULATORS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2014-10-30 WO disclosed