SCHEMBL16200081

SCHEMBL16200081

COc1ccc(-c2c(Cl)c(C)nn2C)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.45
CNR1 P21554 2/20 0.44
CNR2 P34972 1/20 0.44
GPR55 Q9Y2T6 1/20 0.44
ATM Q13315 1/20 0.43
ALDH1A1 P00352 4/20 0.42
LMNA P02545 2/20 0.42
TGFBR1 P36897 1/20 0.42
MAPK14 Q16539 1/20 0.42
MAOA P21397 1/20 0.42
KDM4C Q9H3R0 1/20 0.42
GRM5 P41594 1/20 0.41
NR3C1 P04150 1/20 0.41
PTGS2 P35354 3/20 0.40
KDM4E B2RXH2 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
NPC1 O15118 2/20 0.40
HPGD P15428 2/20 0.40
RAB9A P51151 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14996606 0.83 GRM5 (0.48) BACE1ATMALDH1A1LMNATGFBR1
SCHEMBL16200256 0.82 L3MBTL1 (0.45) CNR1CNR2GPR55ALDH1A1LMNA
SCHEMBL14139215 0.81 ALDH1A1 (0.46) ALDH1A1LMNAMAPK14NR3C1KDM4E
SCHEMBL12856308 0.80 GRM5 (0.46) BACE1CNR1CNR2ATMALDH1A1
SCHEMBL13739115 0.80 ALDH1A1 (0.55) CNR1CNR2ATMALDH1A1LMNA
SCHEMBL13066526 0.79 SLC34A1 (0.51) GRM5
SCHEMBL16200248 0.79 ALDH1A1 (0.40) ALDH1A1LMNAPTGS2KDM4EKMT2A
SCHEMBL12859331 0.78 ATM (0.41) BACE1ATMALDH1A1LMNATGFBR1
SCHEMBL12871642 0.78 KDM4E (0.42) BACE1ATMALDH1A1LMNAKDM4C
SCHEMBL14996631 0.77 MEN1 (0.43) CNR1CNR2GPR55ATMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed