SCHEMBL16200281

SCHEMBL16200281

Cc1c(Cl)c(N2CCCC2=O)nn1C

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.42
POLB P06746 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.39
ALDH1A1 P00352 1/20 0.38
BRD4 O60885 1/20 0.37
BRD2 P25440 1/20 0.37
HSD17B10 Q99714 1/20 0.36
HPGD P15428 1/20 0.35
LMNA P02545 1/20 0.34
CNR2 P34972 1/20 0.34
PDE10A Q9Y233 5/20 0.34
PIP4K2A P48426 1/20 0.33
MEN1 O00255 1/20 0.33
TSHR P16473 1/20 0.33
KMT2A Q03164 1/20 0.33
SIGMAR1 Q99720 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13184168 0.80 L3MBTL1 (0.36) PKMPOLBL3MBTL1ALDH1A1BRD4
SCHEMBL14043925 0.74 PKM (0.42) PKML3MBTL1BRD4BRD2HSD17B10
SCHEMBL16200129 0.71 L3MBTL1 (0.39) L3MBTL1BRD4BRD2HSD17B10HPGD
SCHEMBL18282502 0.71 PKM (0.38) PKML3MBTL1BRD4BRD2HSD17B10
SCHEMBL10274571 0.69 PKM (0.46) PKML3MBTL1BRD4BRD2HSD17B10
SCHEMBL19795212 0.65 DDB1 (0.65) PKMALDH1A1BRD4HSD17B10HPGD
SCHEMBL15081338 0.65 DDB1 (0.52) PKMALDH1A1HSD17B10HPGDLMNA
SCHEMBL13184318 0.65 PDE1A (0.38) PKML3MBTL1BRD4BRD2HSD17B10
SCHEMBL16698832 0.65 MEN1 (0.42) PKML3MBTL1ALDH1A1BRD4BRD2
SCHEMBL17473548 0.65 HSD17B10 (0.43) PKML3MBTL1ALDH1A1BRD4BRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed