SCHEMBL16200322

SCHEMBL16200322

Cc1[nH]nc(-c2cc[nH]n2)c1Cl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.35
IDO1 P14902 1/20 0.32
IKBKB O14920 1/20 0.32
MAP3K14 Q99558 1/20 0.32
ALOX12 P18054 3/20 0.31
MAPT P10636 3/20 0.31
NPSR1 Q6W5P4 3/20 0.31
MEN1 O00255 2/20 0.31
CYP1A2 P05177 2/20 0.31
CYP3A4 P08684 2/20 0.31
CYP2D6 P10635 2/20 0.31
CYP2C9 P11712 2/20 0.31
CYP2C19 P33261 2/20 0.31
KMT2A Q03164 2/20 0.31
GPR55 Q9Y2T6 2/20 0.31
HSP90AA1 P07900 1/20 0.31
KDM4E B2RXH2 1/20 0.31
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3223552 0.71 LRRK2 (0.51) CYP1A2KMT2AKDM4ETDP1MAPK1
SCHEMBL3463988 0.71 TGFBR1 (0.50) HCAR2MAPK1
SCHEMBL16200328 0.71 HCAR2 (0.33) HCAR2IKBKBMAP3K14ALOX12MAPT
SCHEMBL13184423 0.70 ALDH1A1 (0.45) MAPTNPSR1GAAHTTLMNA
SCHEMBL3464248 0.70 CCR1 (0.52) HCAR2MEN1CYP3A4KMT2AHSP90AA1
SCHEMBL3464623 0.70 MAPK14 (0.41)
SCHEMBL13033939 0.68 IKBKB (0.37) IDO1IKBKB
SCHEMBL3464192 0.68 LRRK2 (0.43) MAPK1
SCHEMBL16200111 0.68 HCAR2 (0.33) HCAR2IDO1
SCHEMBL1673128 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed