SCHEMBL16200330

SCHEMBL16200330

Cc1[nH]nc(-c2ccns2)c1Cl

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.33
CYP1A2 P05177 2/20 0.31
CYP3A4 P08684 2/20 0.31
CYP2D6 P10635 2/20 0.31
IKBKB O14920 1/20 0.30
MAP3K14 Q99558 1/20 0.30
GYS1 P13807 1/20 0.30
MEN1 O00255 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30
CYP2C9 P11712 1/20 0.30
ALOX15 P16050 1/20 0.30
ALOX12 P18054 1/20 0.30
MAPK1 P28482 1/20 0.30
CYP2C19 P33261 1/20 0.30
HTT P42858 1/20 0.30
KMT2A Q03164 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
GPR55 Q9Y2T6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16200324 0.66 HCAR2 (0.33) HCAR2CYP1A2CYP3A4CYP2D6IKBKB
SCHEMBL3223552 0.66 LRRK2 (0.51) CYP1A2ALOX15MAPK1KMT2A
SCHEMBL16200204 0.64 NPC1 (0.38) CYP1A2MEN1MAPTCYP2C9MAPK1
SCHEMBL3464248 0.64 CCR1 (0.52) HCAR2CYP3A4MEN1MAPK1KMT2A
SCHEMBL3465575 0.64 MAPK1 (0.47) MAPK1
SCHEMBL3464003 0.64 MAP2K4 (0.55) CYP1A2CYP3A4
SCHEMBL3464623 0.64 MAPK14 (0.41)
SCHEMBL16200322 0.64 HCAR2 (0.35) HCAR2CYP1A2CYP3A4CYP2D6IKBKB
SCHEMBL24119890 0.63 ERBB2 (0.45) CYP1A2CYP3A4CYP2D6IKBKBMAP3K14
SCHEMBL16200197 0.62 CYP11B2 (0.38) MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed