SCHEMBL16201140

SCHEMBL16201140

COC(=O)C[C@H](NC(=O)C1CCC(F)(F)CC1)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 13/20 0.52
KCNH2 Q12809 3/20 0.49
CYP3A4 P08684 1/20 0.49
ADRA2A P08913 1/20 0.49
CYP2C9 P11712 1/20 0.49
KCNE1 P15382 1/20 0.49
OPRM1 P35372 1/20 0.49
KCNQ1 P51787 1/20 0.49
SLC47A1 Q96FL8 1/20 0.49
ITGB3 P05106 1/20 0.48
ITGA2B P08514 1/20 0.48
KCNQ3 O43525 2/20 0.48
KCNQ2 O43526 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
RECQL P46063 1/20 0.47
KCNQ4 P56696 1/20 0.43
KCNQ5 Q9NR82 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5142094 0.90 CCR5 (0.52) CCR5KCNH2CYP3A4ADRA2ACYP2C9
SCHEMBL13714450 0.90 CCR5 (0.52) CCR5KCNH2CYP3A4ADRA2ACYP2C9
SCHEMBL4130344 0.88 CCR5 (0.54) CCR5KCNH2CYP3A4ADRA2ACYP2C9
SCHEMBL14420637 0.88 CCR5 (0.54) CCR5KCNH2CYP3A4ADRA2ACYP2C9
SCHEMBL14218307 0.88 ITGB3 (0.60) CCR5KCNH2CYP3A4ADRA2ACYP2C9
SCHEMBL3882540 0.88 ITGB3 (0.60) CCR5KCNH2CYP3A4ADRA2ACYP2C9
SCHEMBL14416420 0.87 CCR5 (0.53) CCR5KCNH2CYP3A4ADRA2ACYP2C9
SCHEMBL1573757 0.86 RECQL (0.59) CCR5KCNH2ITGB3ITGA2BSMN1; SMN2
SCHEMBL1573959 0.86 RECQL (0.59) CCR5KCNH2ITGB3ITGA2BSMN1; SMN2
SCHEMBL22904305 0.84 KCNQ3 (0.65) CCR5KCNH2CYP3A4ADRA2ACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014173375-A1 A PROCESS FOR THE SYNTHESIS OF MARAVIROC ZENTIVA, K.S. (CZ) 2014-10-30 WO disclosed