SCHEMBL16207708

SCHEMBL16207708

CNC1(C(=O)N2CCNCC2)CCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.46
KMT2A Q03164 3/20 0.46
KDM4E B2RXH2 1/20 0.46
CA2 P00918 2/20 0.41
CHKA P35790 1/20 0.41
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA9 Q16790 1/20 0.38
CYP1A2 P05177 2/20 0.38
CHRNB2 P17787 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
CHRNB3 Q05901 1/20 0.36
CHRNA6 Q15825 1/20 0.36
POLB P06746 1/20 0.36
EPHX2 P34913 1/20 0.36
PARP1 P09874 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM3 P20309 1/20 0.34
MEN1 O00255 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11937915 0.95 KMT2A (0.44) HSD11B1KMT2AKDM4ECA2CHKA
SCHEMBL16207687 0.93 KDM4E (0.48) HSD11B1KMT2AKDM4ECA2CHKA
SCHEMBL11937897 0.79 MEN1 (0.47) HSD11B1KMT2APOLBMEN1
SCHEMBL13077840 0.79 MEN1 (0.47) HSD11B1KMT2APOLBMEN1
SCHEMBL14473297 0.79 KDM4E (0.51) HSD11B1KMT2AKDM4ECYP1A2EPHX2
SCHEMBL11930102 0.78 CYP1A2 (0.42) HSD11B1KMT2ACA2CHKACA12
SCHEMBL13222588 0.77 CA2 (0.41) HSD11B1KMT2ACA2CHKACA12
SCHEMBL12187920 0.77 CA2 (0.41) HSD11B1KMT2ACA2CHKACA12
SCHEMBL13817707 0.76 HSD11B1 (0.43) HSD11B1KMT2ACYP1A2EPHX2PARP1
SCHEMBL14389589 0.76 L3MBTL3 (0.45) KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2799435-B1 POLY (ADP-RIBOSE) POLYMERASE INHIBITOR CHENGDU DIAO PHARMACEUTICAL GROUP CO LTD (CN) 2018-03-28 EP disclosed
CN-103130723-B Poly (aenosine diphosphate glucose pyrophospheralase (ADP)-ribose) polymerase inhibitor CHENGDU DIAO PHARMACEUTICAL GROUP CO LTD 2015-01-14 CN disclosed
EP-2799435-A1 POLY (ADP-RIBOSE) POLYMERASE INHIBITOR Chengdu Di'ao Pharmaceutical Group Co. Ltd. (CN) 2014-11-05 EP disclosed