SCHEMBL16212943

SCHEMBL16212943

Brc1ccn2cc(C3=COC=C(C4=CC=CCC4)O3)nc2c1

nearest known ligand 0.34

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16212740 0.85 TLR9 (0.46)
SCHEMBL6390141 0.84 RAB9A (0.38) KDM4ENPC1RAB9A
SCHEMBL16212728 0.81 SUV39H2 (0.40)
SCHEMBL16212585 0.80 SUV39H2 (0.37)
SCHEMBL16212479 0.77 SUV39H2 (0.41)
SCHEMBL5308528 0.76 RAB9A (0.45) KDM4ENPC1RAB9A
SCHEMBL2127673 0.72 ALDH1A1 (0.46) KDM4ENPC1RAB9A
SCHEMBL4828410 0.67
SCHEMBL7238218 0.66 MAPT (0.31) NPC1RAB9A
SCHEMBL3584562 0.65 NUDT1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2991983-A1 2-PHENYL OR 2-HETARYL IMIDAZOL[1,2-a]PYRIDINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2016-03-09 EP disclosed
WO-2014177458-A1 2-PHENYL OR 2-HETARYL IMIDAZOL[1,2-a]PYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2014-11-06 WO disclosed