SCHEMBL16213009

SCHEMBL16213009

O=C(O)[C@H](CN1C(=O)C=CC1=O)N1C(=O)CCC1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.53
PKM P14618 1/20 0.53
PTGS1 P23219 5/20 0.35
PTGS2 P35354 5/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 2/20 0.34
KDM4E B2RXH2 1/20 0.34
TP53 P04637 1/20 0.34
GLA P06280 1/20 0.34
POLB P06746 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
ALOX12 P18054 1/20 0.34
NFKB1 P19838 1/20 0.34
APEX1 P27695 1/20 0.34
MAPK1 P28482 1/20 0.34
HSD17B10 Q99714 1/20 0.34
DNMT1 P26358 4/20 0.34
SLC1A2 P43004 1/20 0.34
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL870114 1.00 ALDH1A1 (0.53) ALDH1A1PKMPTGS1PTGS2GAA
SCHEMBL10421278 0.85 ALDH1A1 (0.54) ALDH1A1PKMGAAHPGDKDM4E
SCHEMBL4429188 0.83 ALDH1A1 (0.50) ALDH1A1PKMPTGS1PTGS2HPGD
SCHEMBL502079 0.80 PTGS1 (0.47) ALDH1A1PKMPTGS1PTGS2HPGD
SCHEMBL4738905 0.79 PTGS1 (0.50) ALDH1A1PKMPTGS1PTGS2HPGD
SCHEMBL5162325 0.76 ALDH1A1 (0.56) ALDH1A1PKMPTGS1PTGS2GAA
SCHEMBL21620435 0.75 MGLL (0.53) ALDH1A1PKMPTGS1PTGS2HPGD
SCHEMBL31005834 0.75 MGLL (0.53) ALDH1A1PKMPTGS1PTGS2HPGD
SCHEMBL3505155 0.74 ALDH1A1 (0.58) ALDH1A1PKMGAAHPGDKDM4E
SCHEMBL24300565 0.72 ALDH1A1 (0.56) ALDH1A1PKMGAAHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2992008-A1 THERAPEUTIC PEPTIDES GlaxoSmithKline Intellectual Property Development Limited (GB) 2016-03-09 EP disclosed
WO-2014178018-A1 THERAPEUTIC PEPTIDES GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2014-11-06 WO disclosed