SCHEMBL16213867

SCHEMBL16213867

CC(C)(C)OC(=O)C1C2CCC(CC2)[C@H]1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.38
BTK Q06187 1/20 0.38
ALDH1A1 P00352 2/20 0.36
GPR119 Q8TDV5 1/20 0.36
PPM1B O75688 2/20 0.36
PTPN1 P18031 2/20 0.36
PPP1CC P36873 1/20 0.36
KMT2A Q03164 1/20 0.36
MAPK1 P28482 1/20 0.35
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
PREP P48147 3/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6121092 0.92 ALDH1A1 (0.44) HRH3BTKALDH1A1KMT2ALMNA
SCHEMBL21159154 0.92 ALDH1A1 (0.44) HRH3BTKALDH1A1KMT2ALMNA
SCHEMBL2303235 0.83 BTK (0.38) HRH3BTKGPR119MAPK1CHRM2
SCHEMBL12968568 0.83 CHRM2 (0.40) HRH3BTKALDH1A1GPR119KMT2A
SCHEMBL6926352 0.83 CHRM2 (0.40) HRH3BTKALDH1A1GPR119KMT2A
SCHEMBL4685379 0.82 BTK (0.39) HRH3BTKGPR119MAPK1CHRM2
SCHEMBL4685375 0.82 CHRM2 (0.36) HRH3BTKALDH1A1GPR119PPM1B
SCHEMBL4685371 0.82 CHRM2 (0.36) HRH3BTKALDH1A1GPR119PPM1B
SCHEMBL15653981 0.82 HRH3 (0.37) HRH3BTKGPR119PPM1BPTPN1
SCHEMBL30171988 0.81 HRH3 (0.41) HRH3BTKALDH1A1GPR119PPM1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8877775-B2 Substituted 2-aza-bicyclo[2.2.2]octane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin C BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-11-04 US disclosed
US-8877775-B2 Substituted 2-aza-bicyclo[2.2.2]octane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin C BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-11-04 US disclosed