SCHEMBL16214740

SCHEMBL16214740

O=C1NCC2(CC[C@@H](C(=O)OCc3ccccc3)C2)O1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.44
LMNA P02545 1/20 0.44
CHRM2 P08172 1/20 0.44
ADRA2A P08913 1/20 0.44
CYP2D6 P10635 1/20 0.44
DRD1 P21728 1/20 0.44
GAA P10253 2/20 0.43
MAPT P10636 1/20 0.43
KMT2A Q03164 1/20 0.43
PKM P14618 1/20 0.43
BACE1 P56817 1/20 0.43
HPGD P15428 1/20 0.42
GLA P06280 1/20 0.40
DDB1 Q16531 1/20 0.39
CRBN Q96SW2 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ELANE P08246 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1666468 0.90 GAA (0.42) TSHRGAAPKMBACE1HPGD
SCHEMBL1812580 0.80 OPRK1 (0.48) TSHRLMNACYP2D6GAAKMT2A
SCHEMBL1665969 0.77 TSHR (0.39) TSHRLMNACHRM2ADRA2ACYP2D6
SCHEMBL6120052 0.76 SMN1; SMN2 (0.46) TSHRLMNAGAAKMT2APKM
SCHEMBL23871646 0.75 ALDH1A1 (0.52) TSHRGAAALDH1A1
SCHEMBL23857529 0.75 ALDH1A1 (0.52) TSHRGAAALDH1A1
SCHEMBL11982109 0.75 LMNA (0.44) TSHRLMNACHRM2ADRA2ACYP2D6
SCHEMBL15457715 0.75 SLC6A2 (0.45) TSHRLMNAGAAKMT2APKM
SCHEMBL3617827 0.75 SLC6A2 (0.45) TSHRLMNAGAAKMT2APKM
SCHEMBL30148934 0.75 ALDH1A1 (0.46) TSHRGAAKMT2APKMBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9221819-B2 Spirocyclic compounds as modulators of chemokine receptor activity BRISTOL-MYERS SQUIBB COMPANY (US) 2015-12-29 US disclosed
US-8877749-B2 Spirocyclic compounds as modulators of chemokine receptor activity Bristol-Myers Squibbs Company (US) 2014-11-04 US disclosed