SCHEMBL16232162

SCHEMBL16232162

O=C(Cl)CC1(c2ccc(F)cc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 15/20 0.60
SLC6A3 Q01959 3/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
SLC6A4 P31645 2/20 0.41
SLC6A2 P23975 1/20 0.41
CACNA1G O43497 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10695332 0.91 HSD11B1 (0.73) HSD11B1SLC6A3SLC6A4SLC6A2CACNA1G
SCHEMBL16232160 0.83 HSD11B1 (0.83) HSD11B1SLC6A3MEN1KMT2A
SCHEMBL17761233 0.81 HSD11B1 (0.60) HSD11B1SLC6A3MEN1KMT2ASLC6A4
SCHEMBL1633828 0.79 HSD11B1 (0.57) HSD11B1SLC6A3MEN1KMT2ASLC6A4
SCHEMBL28271097 0.77 OPRM1 (0.53) HSD11B1SLC6A3
SCHEMBL627571 0.76 HSD11B1 (0.90) HSD11B1SLC6A3MEN1KMT2ASLC6A4
SCHEMBL4245329 0.76 HSD11B1 (0.97) HSD11B1SLC6A3MEN1KMT2ASLC6A4
SCHEMBL17761217 0.75 HSD11B1 (0.66) HSD11B1SLC6A3MEN1KMT2ASLC6A4
SCHEMBL10694536 0.75 SLC6A4 (0.59) HSD11B1SLC6A3SLC6A4SLC6A2
SCHEMBL17761311 0.75 HSD11B1 (0.71) HSD11B1SLC6A3SLC6A4SLC6A2CACNA1G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150299184-A1 Amine Derivatives as Potassium Channel Blockers BIONOMICS LIMITED (AU) 2015-10-22 US disclosed
US-20150299184-A1 Amine Derivatives as Potassium Channel Blockers BIONOMICS LIMITED (AU) 2015-10-22 US disclosed
US-20140336198-A1 Amine Derivatives as Potassium Channel Blockers MERCK PATENT GMBH (DE) 2014-11-13 US disclosed
US-20140336198-A1 Amine Derivatives as Potassium Channel Blockers MERCK PATENT GMBH (DE) 2014-11-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140336198-A1 Amine Derivatives as Potassium Channel Blockers KCNA3, KCNH3, KCNK3 HSD11B1 4199/4885SLC6A3 296/4885MEN1 1902/4885
US-20150299184-A1 Amine Derivatives as Potassium Channel Blockers KCNA3, KCNH3, KCNK3 HSD11B1 4199/4885SLC6A3 296/4885MEN1 1902/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.