SCHEMBL16235149

SCHEMBL16235149

O=CCC(Cc1ccc(Cl)cc1)NC(=O)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 5/20 0.56
ROCK2 O75116 2/20 0.51
PRKACA P17612 2/20 0.51
IRAK1 P51617 2/20 0.51
PRKX P51817 2/20 0.51
ROCK1 Q13464 2/20 0.51
PRKG1 Q13976 2/20 0.51
PKN2 Q16513 2/20 0.51
CLK4 Q9HAZ1 2/20 0.51
RPS6KB1 P23443 1/20 0.51
LIMK1 P53667 1/20 0.51
PRKG2 Q13237 1/20 0.51
HIPK4 Q8NE63 1/20 0.51
AURKB Q96GD4 1/20 0.51
CSNK1G1 Q9HCP0 1/20 0.51
PIN1 Q13526 1/20 0.50
CTSL P07711 1/20 0.49
HTT P42858 1/20 0.49
KDM4E B2RXH2 1/20 0.47
GAA P10253 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL247680 0.76 EPHX1 (0.53) CTRB1MMEMAPK1
SCHEMBL11487694 0.75 CTRB1 (0.71) CTRB1ROCK2PRKACAIRAK1PRKX
SCHEMBL14959409 0.75 MME (0.52) MME
SCHEMBL5685800 0.73 CTRB1 (0.73) CTRB1ROCK2PRKACAIRAK1PRKX
SCHEMBL3682311 0.73 CTRB1 (0.73) CTRB1ROCK2PRKACAIRAK1PRKX
SCHEMBL3682310 0.73 CTRB1 (0.73) CTRB1ROCK2PRKACAIRAK1PRKX
SCHEMBL5262773 0.73 CNR1 (0.72) CNR1CNR2
SCHEMBL11582081 0.72 ROCK2 (0.70) CTRB1ROCK2PRKACAIRAK1PRKX
SCHEMBL11582078 0.72 ROCK2 (0.70) CTRB1ROCK2PRKACAIRAK1PRKX
SCHEMBL12029124 0.72 CTRB1 (0.71) CTRB1ROCK2PRKACAIRAK1PRKX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014184235-A1 BENZAMIDE TRPA1 ANTAGONISTS Acturum Life Science AB (SE) 2014-11-20 WO claimed
WO-2014184235-A1 BENZAMIDE TRPA1 ANTAGONISTS Acturum Life Science AB (SE) 2014-11-20 WO disclosed