SCHEMBL16258183

SCHEMBL16258183

Cc1cc(C(O)C#N)ccc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.44
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
LMNA P02545 3/20 0.34
ESR1 P03372 3/20 0.34
ESR2 Q92731 3/20 0.34
ALDH1A1 P00352 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
ADRB1 P08588 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRB3 P13945 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
GRM5 P41594 1/20 0.33
GAA P10253 1/20 0.32
GFER P55789 1/20 0.32
ALPG P10696 1/20 0.32
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4631294 0.82 TSHR (0.48) TSHRAKR1C3AKR1C2LMNAESR1
SCHEMBL7604782 0.82 TSHR (0.48) TSHRAKR1C3AKR1C2LMNAESR1
SCHEMBL8943569 0.81 CES2 (0.39) TSHRAKR1C3AKR1C2ALDH1A1ADRB1
SCHEMBL4062640 0.78 TSHR (0.44) TSHRLMNAESR1ESR2ALDH1A1
SCHEMBL30965001 0.78 TSHR (0.44) TSHRESR1ESR2ALDH1A1
SCHEMBL8251464 0.76 UGT2B7 (0.45) TSHRAKR1C3AKR1C2LMNATDP1
SCHEMBL12875453 0.75 SLC6A2 (0.46) TSHRLMNAALDH1A1ACHE
SCHEMBL16216180 0.75 PDE2A (0.42) TSHRAKR1C3AKR1C2LMNATDP1
SCHEMBL14154807 0.75 AKR1C3 (0.37) TSHRAKR1C3AKR1C2LMNATDP1
SCHEMBL23429142 0.73 S1PR1 (0.39) ADRA2BS1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2186794-B1 MONOHALOGENATED PYRETHRIC ACID ALPHA-CYANO-4-FLUORO-3-PHENOXYBENZYL ESTER AND ITS PREPARATION METHOD AND USE UNIV EAST CHINA NORMAL (CN) 2014-11-26 EP disclosed