SCHEMBL7604782

SCHEMBL7604782

N#C[C@@H](O)c1ccc(F)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.48
CES2 O00748 2/20 0.46
CES1 P23141 2/20 0.46
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 2/20 0.34
ALPG P10696 1/20 0.34
ADRB1 P08588 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRB3 P13945 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
S1PR3 Q99500 3/20 0.32
GAA P10253 1/20 0.32
PDPK1 O15530 1/20 0.32
S1PR1 P21453 1/20 0.32
MME P08473 1/20 0.31
AKR1C3 P42330 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4631294 1.00 TSHR (0.48) TSHRCES2CES1ESR1ESR2
SCHEMBL16258183 0.82 TSHR (0.44) TSHRCES2CES1ESR1ESR2
SCHEMBL4062640 0.82 TSHR (0.44) TSHRCES2CES1ESR1ESR2
SCHEMBL7205406 0.79 CES2 (0.46) TSHRCES2CES1ESR1ESR2
SCHEMBL3718088 0.77 CES2 (0.39) CES2CES1ESR1ESR2SMN1; SMN2
SCHEMBL11030008 0.76 PDE2A (0.41) TSHR
SCHEMBL6908022 0.76 TSHR (0.60) TSHRESR1ESR2SMN1; SMN2ALDH1A1
SCHEMBL199580 0.76 TSHR (0.60) TSHRESR1ESR2SMN1; SMN2ALDH1A1
SCHEMBL16951204 0.75 CES2 (0.38) CES2CES1ESR1ESR2SMN1; SMN2
SCHEMBL5660658 0.75 CES2 (0.38) CES2CES1ESR1ESR2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0957083-B1 Process for stabilising cyanhydrines DSM FINE CHEM AUSTRIA GMBH (AT) 2002-04-10 EP claimed
US-6031123-A Process for stabilizing cyanohydrins DSM FINE CHEMICALS AUSTRIA GMBH (AT) 2000-02-29 US claimed
US-6417377-B1 Process for preparing enantiomer-enriched amino- and hydroxyfuranones DSM FINE CHEMICALS AUSTRIA NFG GMBH & CO KG (AT) 2002-07-09 US disclosed
US-6225095-B1 REACTING ALDEHYDE OR KETONE DISSOLVED IN AN ORGANIC, WATER-IMMISCIBLE OR SLIGHTLY MISCIBLE DILUENT, AN AQUEOUS HYDROXYNITRILE LYASE SOLUTION, AND A CYANIDE GROUP DONOR TO FORM AN EMULSION WHICH IS MAINTAINED BY STIRRING DSM FINE CHEMICALS AUSTRIA GMBH (AT) 2001-05-01 US disclosed
US-6031123-A Process for stabilizing cyanohydrins DSM FINE CHEMICALS AUSTRIA GMBH (AT) 2000-02-29 US disclosed