SCHEMBL23429142

SCHEMBL23429142

Cc1cc(C(O)c2cccc(C#N)c2)ccc1F

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.39
ADRA1D P25100 4/20 0.36
ADRA1A P35348 2/20 0.36
ADRA2B P18089 1/20 0.36
ENPP2 Q13822 1/20 0.36
GRM4 Q14833 1/20 0.36
ADRA1B P35368 1/20 0.36
GSK3B P49841 1/20 0.35
P4HB P07237 1/20 0.34
CNR1 P21554 5/20 0.34
CNR2 P34972 4/20 0.34
MGLL Q99685 1/20 0.34
MCHR1 Q99705 1/20 0.34
ACLY P53396 1/20 0.34
TNF P01375 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30834043 0.82 GRIN2D (0.38) ADRA1DADRA1AADRA2BENPP2GRM4
SCHEMBL17064633 0.82 GRIN2D (0.38) ADRA1DADRA1AADRA2BENPP2GRM4
SCHEMBL23429078 0.79 ACHE (0.40) CNR2
SCHEMBL1507787 0.77 TSHR (0.48) ENPP2GRM4GSK3BMGLLTNF
SCHEMBL30961611 0.77 TSHR (0.48) ENPP2GRM4GSK3BMGLLTNF
SCHEMBL13714051 0.76 GAA (0.49) S1PR1ENPP2GRM4GSK3BTNF
SCHEMBL17064353 0.74 CA1 (0.45) ADRA1DADRA1AADRA2BENPP2GRM4
SCHEMBL532567 0.73 EGLN2 (0.48)
SCHEMBL16258183 0.73 TSHR (0.44) S1PR1ADRA2B
SCHEMBL4095529 0.72 ENPP2 (0.46) S1PR1ADRA1DADRA1AADRA2BENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3828173-A1 SUBSTITUTED PYRAZOLES AS HUMAN PLASMA KALLIKREIN INHIBITORS BioCryst Pharmaceuticals, Inc. (US) 2021-06-02 EP disclosed