SCHEMBL1626459

SCHEMBL1626459

O=S(=O)(c1ccc(C2CCCCC2)cc1)C(C1CCNCC1)N1CCc2ccccc2C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 3/20 0.42
PRMT5 O14744 2/20 0.41
WDR77 Q9BQA1 1/20 0.41
DRD3 P35462 1/20 0.40
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.39
AKR1C3 P42330 1/20 0.39
NAMPT P43490 1/20 0.39
APOBEC3A P31941 1/20 0.38
APOBEC3G Q9HC16 1/20 0.38
MEN1 O00255 5/20 0.37
KMT2A Q03164 5/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
DPP8 Q6V1X1 1/20 0.36
TSHR P16473 3/20 0.36
NPSR1 Q6W5P4 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MCOLN2 Q8IZK6 1/20 0.36
MCOLN3 Q8TDD5 1/20 0.36
MCOLN1 Q9GZU1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5922605 0.99 HTR6 (0.41) HTR6PRMT5WDR77DRD3LMNA
SCHEMBL1626463 0.89 PRMT5 (0.43) HTR6PRMT5WDR77LMNAHTT
Hydrochloric Acid SCHEMBL5922613 0.88 PRMT5 (0.42) HTR6PRMT5WDR77LMNAHTT
Hydrochloric Acid SCHEMBL14237064 0.86 MEN1 (0.43) HTR6DRD3LMNAAKR1C3MEN1
SCHEMBL14236984 0.78 HTR6 (0.42) HTR6DRD3LMNAMEN1KMT2A
SCHEMBL14237121 0.78 MAPT (0.43) HTR6DRD3LMNAHTTMEN1
SCHEMBL14237108 0.78 MEN1 (0.53) LMNAHTTMEN1KMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL1627341 0.78 HTR6 (0.41) HTR6DRD3LMNAMEN1KMT2A
SCHEMBL14236969 0.77 SMN1; SMN2 (0.43) HTR6LMNAHTTSMN1; SMN2TSHR
Hydrochloric Acid SCHEMBL1625092 0.77 MAPT (0.42) HTR6DRD3LMNAHTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831195-B1 5-HT7 RECEPTOR ANTAGONISTS ESTEVE LABOR DR (ES) 2012-12-19 EP claimed
US-7928121-B2 2-[1-(5-Chloro-2,4-difluoro-benzenesulfonyl)-piperidin-4-ylmethyl]-1,2,3,4-tetrahydroisoquinolinehydrochloride; antidepressant, anxiolytic, hypotensive agent; psychosis, schizophrenia, migraine, cognition activity; pharmacokinetics LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2011-04-19 US disclosed