SCHEMBL16289869

SCHEMBL16289869

O=C(O)Oc1c(CS(=O)(=O)c2ccccc2)ccc2c1ncc1occc12

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.32
KCNA3 P22001 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
MPO P05164 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
KEAP1 Q14145 1/20 0.31
NFE2L2 Q16236 1/20 0.31
ALOX5AP P20292 1/20 0.31
HSD11B1 P28845 1/20 0.30
CYP1A1 P04798 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP1B1 Q16678 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL436372 0.85 TSHR (0.33) ADORA2APTGDR2MPOALDH1A1MAPT
SCHEMBL434274 0.82 SLC40A1 (0.35) ALDH1A1MAPTKEAP1NFE2L2CYP1A1
SCHEMBL16289961 0.75 MAOA (0.34) ALDH1A1MAPTNPSR1KEAP1NFE2L2
SCHEMBL18784225 0.70 G6PD (0.40) MAPTKEAP1NFE2L2
SCHEMBL16289748 0.67 NPC1 (0.31) ALDH1A1
SCHEMBL436444 0.66 KDM4E (0.42) ALDH1A1MAPTNPSR1
SCHEMBL16289891 0.66 MAPT (0.31) ALDH1A1MAPT
SCHEMBL434719 0.62 TSHR (0.35) ALDH1A1MAPTNPSR1
SCHEMBL18784226 0.62 KMT2A (0.46) ALDH1A1KEAP1NFE2L2HSD11B1
SCHEMBL27867868 0.61 G6PD (0.41) KEAP1NFE2L2HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595988-B1 TRICYCLIC COMPOUNDS AND METHDS OF MAKING AND USING SAME ZAFGEN INC (US) 2014-12-17 EP claimed