SCHEMBL1630447

SCHEMBL1630447

O=C(COCc1ccccc1)c1ccc(OCc2ccccc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A1 P22736 1/20 0.68
NR4A2 P43354 1/20 0.68
NR4A3 Q92570 1/20 0.68
MAOB P27338 1/20 0.64
PARP10 Q53GL7 1/20 0.64
PLA2G4B P0C869 1/20 0.63
SRD5A2 P31213 1/20 0.62
EGFR P00533 4/20 0.61
RAB9A P51151 3/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
MAPK1 P28482 2/20 0.59
NPC1 O15118 1/20 0.59
ALDH1A1 P00352 2/20 0.58
MAPT P10636 2/20 0.58
GAA P10253 1/20 0.58
HTT P42858 1/20 0.58
L3MBTL1 Q9Y468 2/20 0.57
LMNA P02545 2/20 0.56
CYP1A2 P05177 1/20 0.56
PTGS1 P23219 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1962776 0.87 MAOB (0.52) NR4A1NR4A2NR4A3MAOBPARP10
SCHEMBL9787125 0.87 PLA2G4B (0.67) NR4A1NR4A2NR4A3MAOBPARP10
SCHEMBL657234 0.86 TDP1 (0.55) RAB9ASMN1; SMN2MAPK1NPC1ALDH1A1
SCHEMBL10797162 0.86 MAOB (0.67) NR4A1NR4A2NR4A3MAOBPARP10
SCHEMBL9653413 0.86 NPC1 (0.65) MAOBRAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL8081324 0.86 NR4A2 (0.57) NR4A1NR4A2NR4A3MAOBPARP10
SCHEMBL9047885 0.86 NR4A1 (0.57) NR4A1NR4A2NR4A3MAOBPARP10
SCHEMBL6899078 0.84 NR4A1 (0.56) NR4A1NR4A2NR4A3MAOBPARP10
SCHEMBL11290489 0.84 EGFR (0.66) NR4A1NR4A2NR4A3MAOBPARP10
SCHEMBL6893992 0.83 NR4A1 (0.55) NR4A1NR4A2NR4A3MAOBPARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 41 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109020883-B 3-cyano-2-aminopyridine derivative and preparation method and application thereof 广西民族大学 2022-02-08 CN claimed
EP-0728128-B1 SUBSTITUTED PHENYL COMPOUNDS RHONE POULENC RORER LTD (GB) 1998-09-16 EP claimed
EP-0728128-A1 SUBSTITUTED PHENYL COMPOUNDS RHONE-POULENC RORER LIMITED (GB) 1996-08-28 EP claimed
WO-1995013262-A1 SUBSTITUTED PHENYL COMPOUNDS RHONE-POULENC RORER LIMITED (GB) 1995-05-18 WO claimed
US-12227472-B2 Series of skin-whitening (lightening) compounds UNIGEN, INC. (US) 2025-02-18 US disclosed
US-20230399282-A1 Series of Skin-Whitening (Lightening) Compounds UNIGEN, INC. (US) 2023-12-14 US disclosed
US-11739040-B2 Series of skin-whitening (lightening) compounds UNIGEN, INC. (US) 2023-08-29 US disclosed
EP-4046619-A1 SERIES OF SKIN-WHITENING (LIGHTENING) COMPOUNDS Unigen, Inc. (US) 2022-08-24 EP disclosed
CN-109020883-B 3-cyano-2-aminopyridine derivative and preparation method and application thereof 广西民族大学 2022-02-08 CN disclosed
EP-3542780-B1 SERIES OF SKIN-WHITENING (LIGHTENING) COMPOUNDS UNIGEN INC (US) 2022-01-19 EP disclosed
US-20210188751-A1 Series of Skin-Whitening (Lightening) Compounds UNIGEN, INC. (US) 2021-06-24 US disclosed
US-10941098-B2 Series of skin whitening (lightening) compounds UNIGEN, INC. (US) 2021-03-09 US disclosed
US-6211234-B1 BENZONITRILE COMPOUNDS WITH ETHER AND SULFIDE GROUPS WITH CARBOXY ACID RHONE-POULENC RORER LIMITED (GB) 2001-04-03 US disclosed
EP-0728128-B1 SUBSTITUTED PHENYL COMPOUNDS RHONE POULENC RORER LTD (GB) 1998-09-16 EP disclosed
EP-0728128-A1 SUBSTITUTED PHENYL COMPOUNDS RHONE-POULENC RORER LIMITED (GB) 1996-08-28 EP disclosed
WO-1995013262-A1 SUBSTITUTED PHENYL COMPOUNDS RHONE-POULENC RORER LIMITED (GB) 1995-05-18 WO disclosed
WO-1992012981-A1 SUBSTITUTED PHENYL-1,3 DIOXOLOQUINOLINE DERIVATIVES AND THEIR USE AS ANTITUMOR AGENTS GLAXO INC. (US) 1992-08-06 WO disclosed
EP-0496634-A1 Substituted phenyl-1,3-dioxoloquinoline derivatives and their use as antitumor agents GLAXO INC. (US) 1992-07-29 EP disclosed
US-5126351-A Inhibitors of topoisomerase GLAXO INC. (US) 1992-06-30 US disclosed
US-3952021-A α-(3,4-Dimethoxyphenethylaminomethyl)-3,4 or 3,5-dihydroxybenzylalcohols and salts thereof TANABE SEIYAKU CO., LTD. (JA) 1976-04-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11739040-B2 Series of skin-whitening (lightening) compounds TYR, TH, MAOB NR4A1 2772/4885NR4A2 1977/4885NR4A3 2134/4885
US-20230399282-A1 Series of Skin-Whitening (Lightening) Compounds TYR, TH, MAOB NR4A1 2772/4885NR4A2 1977/4885NR4A3 2134/4885
US-10941098-B2 Series of skin whitening (lightening) compounds TYR, MAOB, TH NR4A1 2962/4885NR4A2 2178/4885NR4A3 2251/4885
US-20210188751-A1 Series of Skin-Whitening (Lightening) Compounds TYR, TH, MAOB NR4A1 2772/4885NR4A2 1977/4885NR4A3 2134/4885
US-12227472-B2 Series of skin-whitening (lightening) compounds TYR, TH, MAOB NR4A1 2772/4885NR4A2 1977/4885NR4A3 2134/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.