SCHEMBL16314531

SCHEMBL16314531

CNCC(O)COc1ccc(N)cc1

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA12 O43570 8/20 0.64
CA1 P00915 8/20 0.64
CA2 P00918 8/20 0.64
CA9 Q16790 8/20 0.64
KDM4E B2RXH2 1/20 0.56
ADRB1 P08588 8/20 0.56
ADRB2 P07550 7/20 0.56
ADRB3 P13945 2/20 0.56
PTGS1 P23219 1/20 0.51
SLC6A2 P23975 1/20 0.51
ALOX15 P16050 1/20 0.51
MAPT P10636 2/20 0.50
HTT P42858 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
CYP2D6 P10635 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22640129 0.84 KDM4E (0.71) CA12CA1CA2CA9KDM4E
SCHEMBL22639981 0.84 KDM4E (0.71) CA12CA1CA2CA9KDM4E
SCHEMBL6259021 0.84 CA12 (0.61) CA12CA1CA2CA9KDM4E
SCHEMBL5390387 0.83 PTGS1 (0.74) KDM4EADRB1ADRB2ADRB3PTGS1
SCHEMBL13357760 0.83 ADRB3 (0.60) CA12CA1CA2CA9KDM4E
SCHEMBL7934862 0.83 MAPT (0.55) CA1CA2CA9KDM4EADRB1
SCHEMBL5354594 0.83 CA12 (0.60) CA12CA1CA2CA9KDM4E
SCHEMBL16090435 0.82 ADRB1 (0.70) CA12CA1CA2CA9KDM4E
SCHEMBL6262690 0.82 ADRB1 (0.70) CA12CA1CA2CA9KDM4E
SCHEMBL6786842 0.82 ADRB2 (0.59) ADRB1ADRB2ADRB3PTGS1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2298304-A2 Carboline derivatives useful in the treatment of cancer PTC Therapeutics, Inc. (US) 2011-03-23 EP disclosed