SCHEMBL16319144

SCHEMBL16319144

CC(C)(C)OC(=O)ON1CC2=C(C1)CN(C(=O)c1ccccc1C(F)(F)F)C2

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPY2R P49146 2/20 0.44
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
HTR2B P41595 1/20 0.42
MAPK14 Q16539 1/20 0.42
SCD O00767 4/20 0.41
MGLL Q99685 2/20 0.40
P2RX7 Q99572 2/20 0.39
GBA1 P04062 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7934516 0.86 NPY2R (0.46) NPY2RCYP2C9CYP2C19HTR2BMAPK14
SCHEMBL518633 0.78 CYP2C9 (0.53) CYP2C9CYP2C19HTR2BMAPK14SCD
SCHEMBL25933 0.76 POLB (0.58) NPY2RCYP2C9CYP2C19HTR2BMAPK14
SCHEMBL3402775 0.76 ELANE (0.35)
SCHEMBL27728713 0.74 SCD (0.51) NPY2RCYP2C9CYP2C19HTR2BMAPK14
SCHEMBL1921758 0.74 CYP2C9 (0.49) CYP2C9CYP2C19HTR2BMAPK14SCD
SCHEMBL2818668 0.71 SPR (0.45) NPY2RCYP2C9CYP2C19HTR2BMAPK14
Trifluoroacetic Acid SCHEMBL518486 0.70 CYP2C9 (0.48) CYP2C9CYP2C19HTR2BMAPK14SCD
SCHEMBL2863943 0.70 LMNA (0.51)
SCHEMBL1222761 0.69 SIGMAR1 (0.55) NPY2RCYP2C9CYP2C19HTR2BMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2328898-B1 2-HETEROARYL-PYRROLO[3,4-C]PYRROLE DERIVATIVES AND THEIR USE AS SCD INHIBITORS SANOFI SA (FR) 2014-12-24 EP disclosed