SCHEMBL16319196

SCHEMBL16319196

CC(C)(C)[Si](OCc1cc(C#N)ncn1)(c1ccccc1)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.34
SMYD2 Q9NRG4 2/20 0.33
MAOB P27338 2/20 0.31
GPR119 Q8TDV5 1/20 0.31
CYP3A4 P08684 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
GRM5 P41594 1/20 0.31
GRM1 Q13255 1/20 0.31
KMO O15229 1/20 0.31
GABRA5 P31644 1/20 0.31
CYP19A1 P11511 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16319292 0.80 SMYD2 (0.32) SMYD2CYP3A4HTTSMN1; SMN2GRM5
SCHEMBL1734113 0.73 SMYD2 (0.35) SMYD2CYP3A4HTTSMN1; SMN2CYP19A1
SCHEMBL29623921 0.73 GABRA1 (0.38) SMYD2CYP3A4HTTSMN1; SMN2GRM5
SCHEMBL16318760 0.73 LOXL2 (0.34) SMYD2CYP3A4HTTSMN1; SMN2GRM5
SCHEMBL4147048 0.70 SMYD2 (0.32) SMYD2GABRA5
SCHEMBL1314001 0.70 AGXT (0.42) SMYD2MAOBCYP3A4HTTSMN1; SMN2
SCHEMBL8794941 0.69 MMP3 (0.38) CYP3A4
SCHEMBL3248397 0.69 UHRF1 (0.37) CYP3A4HTTSMN1; SMN2GRM5GRM1
SCHEMBL17288279 0.69 FFAR1 (0.34) SMYD2CYP3A4HTTSMN1; SMN2
SCHEMBL3544323 0.69 PTGER4 (0.33) SMYD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382188-B2 Aromatic ring compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-07-05 US disclosed
EP-2816023-A1 AROMATIC RING COMPOUND Takeda Pharmaceutical Company Limited (JP) 2014-12-24 EP disclosed