SCHEMBL16319407

SCHEMBL16319407

NC(=O)c1cc[c]c(NCC2CCCCC2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.42
PARP15 Q460N3 3/20 0.42
PARP10 Q53GL7 3/20 0.42
OPRD1 P41143 2/20 0.42
CD38 P28907 1/20 0.41
OPRK1 P41145 2/20 0.40
HDAC6 Q9UBN7 4/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
CA2 P00918 1/20 0.39
NAMPT P43490 1/20 0.38
F2 P00734 1/20 0.38
PLG P00747 1/20 0.38
PRSS1 P07477 1/20 0.38
PRSS2 P07478 1/20 0.38
PRSS3 P35030 1/20 0.38
ST14 Q9Y5Y6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16320397 0.79 FAAH (0.44) HDAC6CA2FAAHTRPA1EPHX2
SCHEMBL1238942 0.76 NPC1 (0.50) OPRM1PARP15PARP10OPRD1CD38
SCHEMBL16319711 0.76 NPC1 (0.41) CD38OPRK1KMT2AMEN1NPC1
SCHEMBL5547776 0.73 RXFP1 (0.45) OPRM1OPRK1HDAC6HDAC3HDAC4
SCHEMBL16319993 0.72 TSHR (0.43) KMT2AMEN1NAMPT
SCHEMBL2792642 0.70 CD38 (0.41) PARP15PARP10CD38KMT2AMEN1
SCHEMBL16319436 0.69 MAPK8 (0.42) HDAC6FAAHTRPA1EPHX2FAAH2
SCHEMBL23169493 0.69 JAK2 (0.47) PARP15PARP10CD38HDAC6HDAC3
SCHEMBL4961543 0.68 FAAH (0.59) OPRM1OPRK1HDAC6KMT2AMEN1
SCHEMBL3090215 0.67 HDAC6 (0.71) OPRM1PARP15PARP10OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2544684-B1 4,4-DISUBSTITUTED PIPERIDINE DERIVATIVES USEFUL AS INHIBITORS OF DIPEPTIDYL PEPTIDASE-1 (DPP-1) JANSSEN PHARMACEUTICA NV (BE) 2014-12-24 EP disclosed