SCHEMBL16319982

SCHEMBL16319982

FC(F)(F)c1cc[c]c(OCC2CCCCC2)c1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SCN8A Q9UQD0 2/20 0.40
SCN10A Q9Y5Y9 2/20 0.40
PTGER1 P34995 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
PDK2 Q15119 2/20 0.38
MGLL Q99685 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37
PTGS2 P35354 2/20 0.37
PARP10 Q53GL7 2/20 0.36
PARP15 Q460N3 1/20 0.35
SLC6A4 P31645 1/20 0.35
HTR6 P50406 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13723295 0.81 PARP10 (0.41) MAOAMAOBPARP10PARP15SLC6A4
SCHEMBL15474826 0.79 MAOA (0.48) MAOAMAOBPARP10PARP15
SCHEMBL15474787 0.78 PARP10 (0.40) MAOAMAOBPARP10PARP15SLC6A4
SCHEMBL2376907 0.78 SLC6A4 (0.49) PTGER1MAOAMAOBPARP10PARP15
SCHEMBL13722740 0.76 PARP10 (0.40) PARP10PARP15
SCHEMBL2376749 0.75 SLC6A2 (0.42) MAOAMAOBPTGDR2PARP10PARP15
SCHEMBL160634 0.75 MAPT (0.36) MAOBPTGS2
SCHEMBL21430664 0.74 KMT2A (0.52) PDK2PARP10
SCHEMBL6226618 0.73 L3MBTL1 (0.41) MAOB
SCHEMBL5547776 0.72 RXFP1 (0.45) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2544684-B1 4,4-DISUBSTITUTED PIPERIDINE DERIVATIVES USEFUL AS INHIBITORS OF DIPEPTIDYL PEPTIDASE-1 (DPP-1) JANSSEN PHARMACEUTICA NV (BE) 2014-12-24 EP disclosed