SCHEMBL16334142

SCHEMBL16334142

Cc1cc(C)c(-c2ccc3c(c2)[N]c2cc(-c4c(C)cc(C)cc4C)ccc2-3)c(C)c1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
HSD11B1 P28845 1/20 0.31
SRC P12931 1/20 0.31
PSMB5 P28074 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL815694 0.84 MEN1 (0.33) MEN1ALDH1A1MAPTKMT2ASMN1; SMN2
SCHEMBL339008 0.75 TP53 (0.43) ALDH1A1MAPTESR1ESR2
SCHEMBL5550613 0.74 MEN1 (0.32) MEN1ALDH1A1MAPTKMT2ASMN1; SMN2
SCHEMBL31299941 0.73 TP53 (0.41) ALDH1A1MAPTESR1ESR2
SCHEMBL716719 0.73 MEN1 (0.33) MEN1ALDH1A1MAPTKMT2ASMN1; SMN2
SCHEMBL6382158 0.73 ALDH1A1 (0.40) MEN1ALDH1A1MAPTKMT2ASMN1; SMN2
SCHEMBL27845453 0.72 MEN1 (0.33) MEN1ALDH1A1MAPTKMT2ASMN1; SMN2
SCHEMBL7939919 0.72 MAPT (0.39) MEN1ALDH1A1MAPTKMT2ASMN1; SMN2
SCHEMBL30122516 0.72 ALDH1A1 (0.39) MEN1ALDH1A1MAPTKMT2ASMN1; SMN2
SCHEMBL23537533 0.71 CYP1A2 (0.41) ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3925989-A1 MOLECULAR WEIGHT CONTROL OF POLYOLEFINS USING HALOGENATED BIS-PHENYLPHENOXY CATALYSTS Dow Global Technologies LLC (US) 2021-12-22 EP claimed
EP-3578578-A1 BIS-BIPHENYLPHENOXY CATALYSTS FOR POLYMERIZATION OF LOW MOLECULAR WEIGHT ETHYLENE-BASED POLYMERS Dow Global Technologies Llc (US) 2019-12-11 EP claimed
US-9975975-B2 Bis-biphenylphenoxy catalysts for polymerization of low molecular weight ethylene-based polymers DOW GLOBAL TECHNOLOGIES LLC (US) 2018-05-22 US claimed
EP-3172250-A1 BIS-BIPHENYLPHENOXY CATALYSTS FOR POLYMERIZATION OF LOW MOLECULAR WEIGHT ETHYLENE-BASED POLYMERS Dow Global Technologies Llc (US) 2017-05-31 EP claimed
US-20170137550-A1 BIS-BIPHENYLPHENOXY CATALYSTS FOR POLYMERIZATION OF LOW MOLECULAR WEIGHT ETHYLENE-BASED POLYMERS DOW GLOBAL TECHNOLOGIES LLC 2017-05-18 US claimed
US-9605098-B2 Molecular weight control of polyolefins using halogenated bis-phenylphenoxy catalysts DOW GLOBAL TECHNOLOGIES LLC (US) 2017-03-28 US claimed
EP-3013871-A1 MOLECULAR WEIGHT CONTROL OF POLYOLEFINS USING HALOGENATED BIS-PHENYLPHENOXY CATALYSTS Dow Global Technologies LLC (US) 2016-05-04 EP claimed
US-20160108156-A1 MOLECULAR WEIGHT CONTROL OF POLYOLEFINS USING HALOGENATED BIS-PHENYLPHENOXY CATALYSTS DOW GLOBAL TECHNOLOGIES LLC 2016-04-21 US claimed
WO-2016014749-A1 BIS-BIPHENYLPHENOXY CATALYSTS FOR POLYMERIZATION OF LOW MOLECULAR WEIGHT ETHYLENE-BASED POLYMERS DOW GLOBAL TECHNOLOGIES LLC (US) 2016-01-28 WO claimed
WO-2014210333-A1 MOLECULAR WEIGHT CONTROL OF POLYOLEFINS USING HALOGENATED BIS-PHENYLPHENOXY CATALYSTS DOW GLOBAL TECHNOLOGIES LLC (US) 2014-12-31 WO claimed
WO-2024050359-A1 GROUP III-HALIDE OR LANTHANIDE-HALIDE BIS(PHENYLPHENOXY) METAL−LIGAND COMPLEXES DOW GLOBAL TECHNOLOGIES LLC (US) 2024-03-07 WO disclosed
WO-2024050368-A1 METHOD OF PRODUCING MULTIMODAL POLYETHYLENE USING AT LEAST ONE GROUP III-BASED OR LANTHANIDE-BASED BIPHENYLPHENOXY CATALYST DOW GLOBAL TECHNOLOGIES LLC (US) 2024-03-07 WO disclosed
EP-4332133-A2 GROUP III AND LANTHANIDE BIS-PHENYL-PHENOXY METAL-LIGAND COMPLEXES Dow Global Technologies LLC (US) 2024-03-06 EP disclosed
US-20230183267-A1 GROUP III AND LANTHANIDE BIS-PHENYL-PHENOXY METAL-LIGAND COMPLEXES DOW GLOBAL TECHNOLOGIES LLC (US) 2023-06-15 US disclosed
US-20230133760-A1 GROUP III AND LANTHANIDE BIS-PHENYL-PHENOXY METAL-LIGAND COMPLEXES DOW GLOBAL TECHNOLOGIES LLC (US) 2023-05-04 US disclosed
US-20170267796-A1 FIVE-COORDINATE BIS-PHENYLPHENOXY CATALYSTS FOR THE PREPARATION OF ETHYLENE-BASED POLYMERS DOW GLOBAL TECHNOLOGIES LLC 2017-09-21 US disclosed
EP-3172250-A1 BIS-BIPHENYLPHENOXY CATALYSTS FOR POLYMERIZATION OF LOW MOLECULAR WEIGHT ETHYLENE-BASED POLYMERS Dow Global Technologies Llc (US) 2017-05-31 EP disclosed
US-20170137550-A1 BIS-BIPHENYLPHENOXY CATALYSTS FOR POLYMERIZATION OF LOW MOLECULAR WEIGHT ETHYLENE-BASED POLYMERS DOW GLOBAL TECHNOLOGIES LLC 2017-05-18 US disclosed
WO-2016089935-A1 FIVE-COORDINATE BIS-PHENYLPHENOXY CATALYSTS FOR THE PREPARATION OF ETHYLENE-BASED POLYMERS DOW GLOBAL TECHNOLOGIES LLC (US) 2016-06-09 WO disclosed
WO-2016014749-A1 BIS-BIPHENYLPHENOXY CATALYSTS FOR POLYMERIZATION OF LOW MOLECULAR WEIGHT ETHYLENE-BASED POLYMERS DOW GLOBAL TECHNOLOGIES LLC (US) 2016-01-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170267796-A1 FIVE-COORDINATE BIS-PHENYLPHENOXY CATALYSTS FOR THE PREPARATION OF ETHYLENE-BASED POLYMERS PARG, AP1M1, BZW1 MEN1 1024/4885ALDH1A1 1532/4885MAPT 893/4885
US-20230133760-A1 GROUP III AND LANTHANIDE BIS-PHENYL-PHENOXY METAL-LIGAND COMPLEXES SSB, SOD1, LGALS3 MEN1 1871/4885ALDH1A1 3746/4885MAPT 1303/4885
US-20230183267-A1 GROUP III AND LANTHANIDE BIS-PHENYL-PHENOXY METAL-LIGAND COMPLEXES SSB, SOD1, LGALS3 MEN1 1938/4885ALDH1A1 3777/4885MAPT 1428/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.