SCHEMBL163419

SCHEMBL163419

O=C(O)Nc1cc(N2CCSCC2)cc(COC2CCCCO2)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.37
CREBBP Q92793 2/20 0.34
EP300 Q09472 1/20 0.34
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
CCNA1 P78396 1/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NPY1R P25929 4/20 0.33
KDM4C Q9H3R0 1/20 0.33
GCK P35557 1/20 0.33
ICAM1 P05362 1/20 0.33
SELE P16581 1/20 0.33
CNR2 P34972 2/20 0.32
CNR1 P21554 1/20 0.32
CA12 O43570 2/20 0.32
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL111995 0.89 CNR2 (0.34) KCNH2CREBBPEP300CCNA2CDK2
SCHEMBL3411723 0.82 MEN1 (0.39) CREBBPEP300CCNA2CDK2CCNA1
SCHEMBL962706 0.80 OPRM1 (0.35) KCNH2CREBBPEP300KDM4CGCK
SCHEMBL113428 0.80 KCNH2 (0.36) KCNH2CREBBPEP300NPY1RKDM4C
SCHEMBL113716 0.80 KCNH2 (0.41) KCNH2CREBBPEP300MEN1KMT2A
SCHEMBL113359 0.77 ALOX5AP (0.34) KCNH2CREBBPEP300GCKCNR2
SCHEMBL7014486 0.77 KCNH2 (0.39) KCNH2CREBBPEP300NPY1RKDM4C
SCHEMBL7016133 0.75 CFTR (0.40) MEN1KMT2AKDM4C
SCHEMBL962329 0.74 HTR2C (0.33)
SCHEMBL3412288 0.74 KDM4C (0.44) CREBBPEP300MEN1KMT2AKDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424860-A1 HETEROARYLTHIOMETHYL PYRIDINE DERIVATIVE MSD K.K. (JP) 2012-03-07 EP disclosed