SCHEMBL7014486

SCHEMBL7014486

C[Si](C)(C)CCOC(=O)Nc1cc(N2CCOCC2)cc(COC2CCCCO2)n1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 9/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
MAPT P10636 1/20 0.38
NPY1R P25929 10/20 0.37
GCK P35557 1/20 0.33
ALDH1A1 P00352 2/20 0.32
EP300 Q09472 1/20 0.32
CREBBP Q92793 1/20 0.32
KDM4C Q9H3R0 1/20 0.32
TP53 P04637 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL113716 0.88 KCNH2 (0.41) KCNH2MAPTNPY1RALDH1A1EP300
SCHEMBL113428 0.82 KCNH2 (0.36) KCNH2NPY1RGCKEP300CREBBP
SCHEMBL962706 0.81 OPRM1 (0.35) KCNH2GCKEP300CREBBPKDM4C
SCHEMBL111995 0.79 CNR2 (0.34) KCNH2NPC1RAB9ANPY1RGCK
SCHEMBL7012955 0.78 KCNH2 (0.35) KCNH2NPY1REP300CREBBP
SCHEMBL113359 0.78 ALOX5AP (0.34) KCNH2GCKEP300CREBBP
SCHEMBL7016133 0.77 CFTR (0.40) KDM4C
SCHEMBL163419 0.77 KCNH2 (0.37) KCNH2NPY1RGCKEP300CREBBP
SCHEMBL7020498 0.76 KCNH2 (0.41) KCNH2SMN1; SMN2NPC1RAB9AMAPT
SCHEMBL114808 0.72 CREBBP (0.36) SMN1; SMN2NPC1RAB9AGCKEP300

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889034-B1 AMINOPYRIDINE DERIVATIVES BANYU PHARMA CO LTD (JP) 2003-09-17 EP disclosed
US-6011039-A USEFUL AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS; TREATING HYPERPHAGIA, OBESITY OR DIABETES BANYU PHARMACEUTICAL CO., LTD. (JP) 2000-01-04 US disclosed
EP-0889034-A1 AMINOPYRIDINE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1999-01-07 EP disclosed