SCHEMBL16353247

SCHEMBL16353247

Cc1ccc(N(c2ccccc2)c2ccc(C=Cc3ccc(/C=C/C(=O)O)cc3)cc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 3/20 0.63
MAPT P10636 3/20 0.55
ALDH1A1 P00352 1/20 0.55
CYP3A4 P08684 1/20 0.55
HPGD P15428 1/20 0.55
HCAR2 Q8TDS4 2/20 0.55
HDAC3 O15379 1/20 0.55
TNKS O95271 1/20 0.55
HDAC4 P56524 1/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC7 Q8WUI4 1/20 0.55
HDAC2 Q92769 1/20 0.55
HDAC10 Q969S8 1/20 0.55
HDAC11 Q96DB2 1/20 0.55
HDAC8 Q9BY41 1/20 0.55
TNKS2 Q9H2K2 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55
HDAC9 Q9UKV0 1/20 0.55
HDAC5 Q9UQL6 1/20 0.55
CYP1B1 Q16678 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16353266 0.95 TRPM8 (0.55) TRPM8MAPTALDH1A1CYP3A4HPGD
SCHEMBL4237337 0.95 TRPM8 (0.55) TRPM8MAPTALDH1A1CYP3A4HPGD
SCHEMBL16353263 0.95 TRPM8 (0.55) TRPM8MAPTALDH1A1CYP3A4HPGD
SCHEMBL17321127 0.94 TRPM8 (0.60) TRPM8MAPTALDH1A1CYP3A4HPGD
SCHEMBL16353227 0.94 TRPM8 (0.57) TRPM8MAPTALDH1A1CYP3A4HPGD
SCHEMBL16353253 0.94 TRPM8 (0.57) TRPM8MAPTALDH1A1CYP3A4HPGD
SCHEMBL16353264 0.92 HCAR2 (0.64) TRPM8MAPTALDH1A1CYP3A4HPGD
SCHEMBL16353257 0.92 HCAR2 (0.64) TRPM8MAPTALDH1A1CYP3A4HPGD
SCHEMBL380761 0.90 HCAR2 (0.67) TRPM8MAPTALDH1A1CYP3A4HPGD
SCHEMBL380760 0.90 HCAR2 (0.67) TRPM8MAPTALDH1A1CYP3A4HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9541848-B2 Electrophotographic photoreceptor Konica Minolta, Inc. (JP) 2017-01-10 US disclosed
US-9304417-B2 Electrophotographic photoreceptor, electrophotographic image forming apparatus and process cartridge Konica Minolta, Inc. (JP) 2016-04-05 US disclosed
US-20150355560-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR Konica Minolta, Inc. (JP) 2015-12-10 US disclosed
US-20140377694-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, ELECTROPHOTOGRAPHIC IMAGE FORMING APPARATUS AND PROCESS CARTRIDGE Konica Minolta, Inc. (JP) 2014-12-25 US disclosed