SCHEMBL16359587

SCHEMBL16359587

CC(C)(C)OC(=O)N1CCC(=O)C2=CC=CC[C@@H]21

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.35
ALDH1A1 P00352 1/20 0.34
NR1H2 P55055 4/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
THRB P10828 1/20 0.33
GPR119 Q8TDV5 1/20 0.33
NR1H3 Q13133 3/20 0.33
UCHL1 P09936 1/20 0.32
HSD11B1 P28845 1/20 0.32
NPC1 O15118 1/20 0.32
EPHX2 P34913 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22109261 0.71 GLA (0.33) ALDH1A1KDM4EMAPTGPR119NPC1
SCHEMBL30900387 0.68 KDM4E (0.34) ALDH1A1NR1H2KDM4EMAPTTHRB
SCHEMBL16224559 0.68 USP2 (0.39) ATMNR1H2KDM4EMAPTTHRB
SCHEMBL2395205 0.68 USP2 (0.39) ATMNR1H2KDM4EMAPTTHRB
SCHEMBL24918232 0.68 USP2 (0.39) ATMNR1H2KDM4EMAPTTHRB
SCHEMBL5420095 0.66 HSD17B10 (0.42) NR1H2KDM4EMAPTTHRBGPR119
SCHEMBL29115999 0.66 NR1H2 (0.50) NR1H2GPR119NR1H3
SCHEMBL642698 0.66 NR1H2 (0.50) NR1H2GPR119NR1H3
SCHEMBL18071798 0.65 MAPT (0.40) ALDH1A1KDM4EMAPTTHRBGPR119
SCHEMBL22820950 0.64 NPC1 (0.38) NR1H2GPR119UCHL1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009052288-A1 SPIRO-CONDENSED 1, 3, 4-THIADIAZOLE DERIVATIVES FOR INHIBITING KSP KINESIN ACTIVITY SCHERING CORPORATION (US) 2009-04-23 WO disclosed