SCHEMBL1636663

SCHEMBL1636663

NC(=S)c1nc[nH]n1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5494345 0.80
SCHEMBL19281540 0.79 GDA (0.31)
SCHEMBL381885 0.76
Hydrochloric Acid SCHEMBL5454883 0.74
SCHEMBL7377426 0.74
SCHEMBL9792943 0.71
SCHEMBL2241163 0.70
SCHEMBL9663668 0.70 P2RX7 (0.30)
SCHEMBL21642922 0.68
Fumaric Acid SCHEMBL35210763 0.67 TSHR (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112689631-A Microbicidal oxadiazole derivatives 先正达农作物保护股份公司 2021-04-20 CN disclosed
CN-107426963-A For agriculture chemistry mixture to be applied to the method and vehicle of field operating area 巴斯夫欧洲公司 2017-12-01 CN disclosed
US-20110265195-A1 UNIQUE ASSOCIATED KAPOSI'S SARCOMA VIRUS SEQUENCES AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2011-10-27 US disclosed
US-7932066-B2 Unique associated kaposi's sarcoma virus sequences and uses thereof THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2011-04-26 US disclosed
US-20090022748-A1 Unique associated Kaposi's sarcoma virus sequences and uses thereof CHANG YUAN 2009-01-22 US disclosed
US-6500663-B1 TREATING A SUBJECT AFFLICTED WITH A KAPOSI'S SARCOMA CAUSED BY KAPOSI'S SARCOMA ASSOCIATED HERPESVIRUS WHICH COMPRISES ADMINISTERING A NUCLEOSIDE ANALOG OR AN ANTISENSE NUCLEIC ACID THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2002-12-31 US disclosed
US-6348586-B1 NUCLEOTIDE SEQUENCE OF HERPES VIRUS; DIAGNOSIS; VACCINES; VIRICIDES; ANTISENSE AGENTS; TRIPLEX OLIGONUCLEOTIDES; THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2002-02-19 US disclosed
US-6183751-B1 VACCINES; DIAGNOSIS; OPEN READING FRAME; GENETIC ENGINEERING THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2001-02-06 US disclosed
US-6150093-A NUCLEOTIDE SEQUENCES PREFERENTIAL FOR HERPES VIRUS ASSOCIATED WITH A CANCER; FOR TREATMENT, DIAGNOSIS AND DETECTION OF AQUIRED IMMUNODEFICIENCY SYNDROME RELATED CANCER THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2000-11-21 US disclosed
US-6093550-A DIAGNOSING KAPOSI'S SARCOMA(KS) ASSOCIATED HERPESVIRUS INFECTION BY CONTACTING A SAMPLE WITH A KS ASSOCIATED HERPESVIRUS ANTIGEN, DETERMINING THE LEVEL OF KS ASSOCIATED HERPESVIRUS ANTIBODY BOUND TO THE ANTIGEN; IMMUNOASSAY KITS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2000-07-25 US disclosed
WO-1997027208-A1 UNIQUE ASSOCIATED KAPOSI'S SARCOMA VIRUS SEQUENCES AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 1997-07-31 WO disclosed
EP-0726708-A1 VIRUS ASSOCIATED MULTIPLE SCLEROSIS: TREATMENTS, PREVENTION AND DIAGNOSIS THEREOF PATHOGENESIS CORPORATION (US) 1996-08-21 EP disclosed
WO-1996015779-A1 UNIQUE ASSOCIATED KAPOSI'S SARCOMA VIRUS SEQUENCES AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 1996-05-30 WO disclosed
WO-1996006159-A1 UNIQUE ASSOCIATED KAPOSI'S SARCOMA VIRUS SEQUENCES AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 1996-02-29 WO disclosed
WO-1995012313-A1 VIRUS ASSOCIATED MULTIPLE SCLEROSIS: TREATMENTS, PREVENTION AND DIAGNOSIS THEREOF PATHOGENESIS CORPORATION (US) 1995-05-11 WO disclosed
US-4056674-A VIRICIDE, BACTERICIDE ICN PHARMACEUTICALS, INC. (US) 1977-11-01 US disclosed
US-3991078-A VIRICIDES ICN PHARMACEUTICALS, INC. (US) 1976-11-09 US disclosed
US-3976545-A WITH NUCLEOSIDE PHOSPHORYLASE AND RIBOSE-1-PHOSPHATE TO FORM 1-B-D-RIBOFURANOSYL ICN PHARMACEUTICALS, INC. (US) 1976-08-24 US disclosed
US-3976545-A WITH NUCLEOSIDE PHOSPHORYLASE AND RIBOSE-1-PHOSPHATE TO FORM 1-B-D-RIBOFURANOSYL ICN PHARMACEUTICALS, INC. (US) 1976-08-24 US disclosed
US-3927216-A 1,2,4-Triazol E-3-carboxamides for inhibiting virus infections VIRATEK, INC., A CORP. OF DE. 1975-12-16 US disclosed