SCHEMBL16370141

SCHEMBL16370141

CC(=NO)c1ccc(C)c(N)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.57
TDP1 Q9NUW8 2/20 0.57
ALDH1A1 P00352 4/20 0.45
CASP1 P29466 1/20 0.45
GFER P55789 3/20 0.44
POLB P06746 1/20 0.44
CASP3 P42574 1/20 0.44
SENP8 Q96LD8 1/20 0.44
SENP7 Q9BQF6 1/20 0.44
SENP6 Q9GZR1 1/20 0.44
RAB9A P51151 3/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP1A2 P05177 1/20 0.43
KDM4E B2RXH2 5/20 0.42
HPGD P15428 4/20 0.42
HTT P42858 3/20 0.42
LMNA P02545 6/20 0.41
KMT2A Q03164 3/20 0.41
NPC1 O15118 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16370140 1.00 MAPT (0.57) MAPTTDP1ALDH1A1CASP1GFER
SCHEMBL24988733 0.84 ALDH1A1 (0.45) MAPTTDP1ALDH1A1GFERPOLB
SCHEMBL6670064 0.81 ALDH1A1 (0.51) MAPTALDH1A1GFERPOLBCASP3
SCHEMBL19859062 0.80 MAPT (0.57) MAPTTDP1ALDH1A1CASP1GFER
SCHEMBL30935544 0.80 MAPT (0.57) MAPTTDP1ALDH1A1CASP1GFER
SCHEMBL14741800 0.80 MAPT (0.57) MAPTTDP1ALDH1A1CASP1GFER
SCHEMBL25100436 0.76 CYP2C19 (0.51) MAPTALDH1A1GFERPOLBCASP3
SCHEMBL16370214 0.76 TDP1 (0.52) MAPTTDP1ALDH1A1CASP1GFER
SCHEMBL16370215 0.76 TDP1 (0.52) MAPTTDP1ALDH1A1CASP1GFER
SCHEMBL18866954 0.75 MAPT (0.61) MAPTTDP1ALDH1A1CASP1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015004481-A1 IMIDAZO-CONDENSED BICYCLES AS INHIBITORS OF DISCOIDIN DOMAIN RECEPTORS (DDRS) ASTEX THERAPEUTICS LIMITED (GB) 2015-01-15 WO disclosed