SCHEMBL16380773

SCHEMBL16380773

CCN1CCN(Cc2ccc(C(N)=O)cc2Cl)CC1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IP6K1 Q92551 3/20 0.56
ALDH1A1 P00352 5/20 0.48
HPGD P15428 1/20 0.48
DUSP3 P51452 1/20 0.48
PTPN5 P54829 1/20 0.48
PTPN11 Q06124 1/20 0.48
DDR1 Q08345 3/20 0.46
KDM4E B2RXH2 1/20 0.44
POLB P06746 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
SIGMAR1 Q99720 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
NPC1 O15118 1/20 0.43
TP53 P04637 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18922209 0.89 ALDH1A1 (0.57) IP6K1ALDH1A1DDR1KDM4EPOLB
SCHEMBL16380731 0.84 KMT2A (0.53) IP6K1ALDH1A1KDM4ELMNAMAPT
SCHEMBL3992921 0.84 IP6K1 (0.52) IP6K1ALDH1A1DDR1KDM4ETP53
SCHEMBL16380631 0.83 GFER (0.49) IP6K1ALDH1A1DUSP3PTPN5PTPN11
SCHEMBL16380724 0.83 ALDH1A1 (0.48) IP6K1ALDH1A1KDM4EPOLBTDP1
SCHEMBL4264923 0.83 CYP2A13 (0.62) IP6K1ALDH1A1HPGDPOLBLMNA
SCHEMBL16380640 0.81 MAPK1 (0.51) ALDH1A1DUSP3KDM4EPOLBTDP1
SCHEMBL3311056 0.80 NR1H2 (0.52) DDR1
SCHEMBL2776747 0.79 ALDH1A1 (0.59) ALDH1A1POLBLMNAMAPTNPC1
SCHEMBL1696442 0.78 SLC6A4 (0.50) KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9670231-B2 Fused tricyclic amide compounds as multiple kinase inhibitors BEIGENE, LTD. (KY) 2017-06-06 US disclosed
WO-2014206344-A1 FUSED TRICYCLIC AMIDE COMPOUNDS AS MULTIPLE KINASE INHIBITORS BEIGENE, LTD. (GB) 2014-12-31 WO disclosed