SCHEMBL16404612

SCHEMBL16404612

Cc1noc(C)c1-c1cccc(F)c1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 16/20 0.62
BRD2 P25440 5/20 0.62
CREBBP Q92793 4/20 0.59
PTGDR2 Q9Y5Y4 1/20 0.54
NPC1 O15118 1/20 0.54
POLB P06746 1/20 0.54
CASP3 P42574 1/20 0.54
RAB9A P51151 1/20 0.54
SENP7 Q9BQF6 1/20 0.54
BRD3 Q15059 1/20 0.51
LMNA P02545 1/20 0.51
CLK4 Q9HAZ1 1/20 0.51
MAP4K4 O95819 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12487 0.82 NPC1 (0.69) BRD4BRD2CREBBPNPC1POLB
SCHEMBL12077969 0.82 BRD4 (0.55) BRD4BRD2CREBBPLMNA
SCHEMBL980536 0.79 MAP4K4 (0.76) BRD4BRD2CREBBPNPC1POLB
SCHEMBL13036108 0.79 BRD4 (0.57) BRD4BRD2CREBBPBRD3
SCHEMBL16246450 0.79 BRD4 (0.62) BRD4BRD2CREBBPNPC1POLB
SCHEMBL9657290 0.79 BRD4 (0.62) BRD4BRD2CREBBPNPC1POLB
SCHEMBL15330867 0.79 BRD4 (0.58) BRD4BRD2CREBBPNPC1POLB
SCHEMBL16404607 0.78 BRD4 (0.66) BRD4BRD2LMNACLK4
SCHEMBL5714189 0.78 BRD4 (0.61) BRD4BRD2CREBBPNPC1POLB
Hydrochloric Acid SCHEMBL1016039 0.78 MAP4K4 (0.73) BRD4BRD2CREBBPNPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2429993-B1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION BOEHRINGER INGELHEIM INT (DE) 2015-01-21 EP disclosed