SCHEMBL16409554

SCHEMBL16409554

C=NC(=O)c1cccc(OCCCC)c1

nearest known ligand 0.68

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PLA2G4B P0C869 3/20 0.60
KMT2A Q03164 3/20 0.57
SMPD1 P17405 3/20 0.57
THRB P10828 2/20 0.56
NR1H4 Q96RI1 2/20 0.54
THRA P10827 1/20 0.52
KAT6A Q92794 2/20 0.51
USP2 O75604 1/20 0.51
MAPK1 P28482 1/20 0.51
MEN1 O00255 2/20 0.49
ADRB2 P07550 2/20 0.49
AKR1C2 P52895 1/20 0.48
AKR1C1 Q04828 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21157003 0.86 KMT2A (0.52) KMT2ANR1H4KAT6AMAPK1MEN1
SCHEMBL11056943 0.83 KMT2A (0.62) PLA2G4BKMT2ASMPD1THRBNR1H4
SCHEMBL7973296 0.83 KAT6A (0.55) PLA2G4BKMT2ASMPD1THRBNR1H4
SCHEMBL7984991 0.82 KAT6A (0.54) PLA2G4BKMT2ASMPD1THRBNR1H4
SCHEMBL1436145 0.81 THRB (0.65) PLA2G4BKMT2ASMPD1THRBNR1H4
SCHEMBL3315904 0.81 KMT2A (0.84) PLA2G4BKMT2ASMPD1NR1H4
SCHEMBL27903063 0.81 KMT2A (0.64) PLA2G4BKMT2ASMPD1THRBNR1H4
SCHEMBL16196481 0.80 SMPD1 (0.74) PLA2G4BKMT2ASMPD1THRBNR1H4
SCHEMBL7765680 0.80 THRB (0.63) PLA2G4BKMT2ASMPD1THRBNR1H4
SCHEMBL15474092 0.80 THRB (0.63) PLA2G4BKMT2ASMPD1THRBNR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014197313-A2 NOVEL COMPOUNDS AND USES THEREOF KALA PHARMACEUTICALS, INC. (US) 2014-12-11 WO disclosed