SCHEMBL16415751

SCHEMBL16415751

O=C(O)NCCc1ccc(O)c(F)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.53
HSD17B10 Q99714 2/20 0.53
KDM4E B2RXH2 1/20 0.53
ALDH1A1 P00352 1/20 0.53
LMNA P02545 1/20 0.53
HPGD P15428 1/20 0.53
PTGS1 P23219 1/20 0.53
BLM P54132 1/20 0.53
HIF1A Q16665 1/20 0.53
ESRRG P62508 1/20 0.52
TRPV1 Q8NER1 2/20 0.47
ERCC1 P07992 1/20 0.47
ERCC4 Q92889 1/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
GAA P10253 1/20 0.46
ALPL P05186 1/20 0.46
APP P05067 1/20 0.44
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20188223 0.87 MAPT (0.53) MAPTHSD17B10KDM4EALDH1A1LMNA
SCHEMBL6420228 0.84 MAPT (0.72) MAPTHSD17B10KDM4EALDH1A1LMNA
SCHEMBL22772331 0.83 MT-CO2 (0.49) ERCC1ERCC4
SCHEMBL6184638 0.81 MAPT (0.58) MAPTHSD17B10KDM4EALDH1A1LMNA
SCHEMBL27944339 0.80 PLK4 (0.55) MAPTHSD17B10KDM4EALDH1A1LMNA
SCHEMBL3627156 0.79 SMN1; SMN2 (0.55) MAPTLMNATRPV1GAACA1
SCHEMBL31354763 0.79 RAB9A (0.44) CA1CA2
SCHEMBL29444602 0.79 ESRRG (0.45) MAPTHSD17B10KDM4EALDH1A1LMNA
SCHEMBL19235667 0.79 ESRRG (0.45) MAPTHSD17B10KDM4EALDH1A1LMNA
SCHEMBL1338001 0.78 KDM4E (0.52) MAPTHSD17B10KDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111051309-B Triazolotriazine derivatives useful as A2A receptor antagonists 浙江春禾医药科技有限公司 2023-05-26 CN disclosed
CN-111051309-A Triazolotriazine derivatives useful as A2A receptor antagonists 浙江春禾医药科技有限公司 2020-04-21 CN disclosed
WO-2015013318-A1 BORON-CONTAINING SMALL MOLECULES ANACOR PHARMACEUTICALS, INC. (US) 2015-01-29 WO disclosed