SCHEMBL164236

SCHEMBL164236

CCCOc1ccc(C#Cc2ccc(CCCNC(=O)OC(C)(C)C)cc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACACB O00763 13/20 0.62
CA12 O43570 5/20 0.54
CA1 P00915 5/20 0.54
CA2 P00918 5/20 0.54
CA9 Q16790 5/20 0.54
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19003451 0.87 ACACB (0.61) ACACBCA12CA1CA2CA9
SCHEMBL17366464 0.83 CA12 (0.59) CA12CA1CA2CA9ALDH1A1
SCHEMBL13907700 0.82 ALDH1A1 (0.68) ACACBCA12CA1CA2CA9
SCHEMBL4656567 0.81 S1PR1 (0.60) CA12CA1CA2CA9
SCHEMBL16234541 0.81 CA12 (0.64) CA12CA1CA2CA9L3MBTL1
SCHEMBL1541945 0.80 CA1 (0.64) ACACBCA12CA1CA2CA9
SCHEMBL13185193 0.80 CA12 (0.67) CA12CA1CA2CA9ALDH1A1
SCHEMBL5015557 0.80 CA1 (0.59) CA12CA1CA2CA9
SCHEMBL910539 0.80 CA1 (0.62) CA12CA1CA2CA9
SCHEMBL3174253 0.80 CA1 (0.53) CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611771-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF Boehringer Ingelheim International GmbH (DE) 2013-07-10 EP disclosed
WO-2012028676-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-03-08 WO disclosed