SCHEMBL16440211

SCHEMBL16440211

CCCCOc1cncc(Cl)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP2D6 P10635 8/20 0.37
CYP3A4 P08684 6/20 0.37
CDK2 P24941 1/20 0.36
CYP2C9 P11712 3/20 0.36
CYP19A1 P11511 2/20 0.36
CYP2C19 P33261 2/20 0.36
CCR4 P51679 1/20 0.35
CYP1A2 P05177 1/20 0.35
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3272531 0.93 CYP3A4 (0.40) NPC1RAB9ASMN1; SMN2HSD17B10CYP2D6
SCHEMBL4437979 0.91 CDK2 (0.38) NPC1RAB9ASMN1; SMN2HSD17B10CYP3A4
SCHEMBL4263969 0.86 CYP2D6 (0.42) NPC1RAB9ASMN1; SMN2HSD17B10CYP2D6
SCHEMBL4434419 0.82 CDK2 (0.40) HSD17B10CYP3A4CDK2CYP2C9CYP19A1
SCHEMBL3267198 0.79 CDK2 (0.38) CDK2HTR2AHTR2CHTR2B
SCHEMBL16631651 0.78 CYP2D6 (0.37) NPC1RAB9ASMN1; SMN2HSD17B10CYP2D6
SCHEMBL3266814 0.76 KCNA3 (0.47) CDK2ALDH1A1
SCHEMBL3268390 0.76 KCNA3 (0.52) SMN1; SMN2CDK2ALDH1A1LMNATSHR
SCHEMBL4268041 0.76 GABRP (0.38) NPC1RAB9ASMN1; SMN2HSD17B10GABRP
SCHEMBL3272371 0.75 KCNA3 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107567443-B Biaryl derivatives as GPR120 agonists 株式会社LG化学 2023-04-28 CN disclosed
CN-115925679-A Biaryl derivatives as GPR120 agonists 株式会社LG化学 2023-04-07 CN disclosed
EP-3239143-B1 BIARYL DERIVATIVE AS GPR120 AGONIST LG CHEMICAL LTD (KR) 2023-03-22 EP disclosed
US-20220135574-A1 BIARYL DERIVATIVE AS GPR120 AGONIST LG CHEM, LTD. (KR) 2022-05-05 US disclosed
US-11261186-B2 Biaryl derivative as GPR120 agonist LG CHEM. LTD. (KR) 2022-03-01 US disclosed
CN-107567443-A biaryl derivatives as GPR120 agonists 株式会社LG化学 2018-01-09 CN disclosed
US-20170349594-A1 BIARYL DERIVATIVE AS GPR120 AGONIST LG CHEM, LTD. (KR) 2017-12-07 US disclosed
EP-3239143-A2 BIARYL DERIVATIVE AS GPR120 AGONIST LG Chem, Ltd. (KR) 2017-11-01 EP disclosed
EP-3027601-B1 SYK INHIBITORS GILEAD SCIENCES INC (US) 2017-10-25 EP disclosed
US-20160368918-A1 SYK INHIBITORS Kronos Bio, Inc. 2016-12-22 US disclosed
US-9376441-B2 Substituted pyrrolidines as SYK inhibitors GILEAD SCIENCES, INC. (US) 2016-06-28 US disclosed
US-20150038488-A1 SYK INHIBITORS Kronos Bio, Inc. 2015-02-05 US disclosed
WO-2015017610-A1 SYK INHIBITORS GILEAD SCIENCES, INC. (US) 2015-02-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220135574-A1 BIARYL DERIVATIVE AS GPR120 AGONIST GPR119, GLP1R, GIPR NPC1 1654/4885RAB9A 2293/4885SMN1; SMN2 3448/4885
US-20150038488-A1 SYK INHIBITORS SYK, BTK, LYN NPC1 4653/4885RAB9A 3263/4885SMN1; SMN2 3200/4885
US-20160368918-A1 SYK INHIBITORS SYK, BTK, LYN NPC1 4638/4885RAB9A 3273/4885SMN1; SMN2 3271/4885
US-20170349594-A1 BIARYL DERIVATIVE AS GPR120 AGONIST GPR119, GLP1R, GIPR NPC1 1654/4885RAB9A 2293/4885SMN1; SMN2 3448/4885
US-11261186-B2 Biaryl derivative as GPR120 agonist GPR119, GPR88, FFAR1 NPC1 640/4885RAB9A 2731/4885SMN1; SMN2 4496/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.