SCHEMBL1644874

SCHEMBL1644874

COc1ccccc1NC(=O)CN(C)C

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.61
MEN1 O00255 2/20 0.61
KMT2A Q03164 2/20 0.61
POLB P06746 2/20 0.61
MAPT P10636 3/20 0.60
HTT P42858 2/20 0.60
GAA P10253 1/20 0.60
MAPK1 P28482 1/20 0.60
LMNA P02545 2/20 0.59
HSD17B10 Q99714 1/20 0.58
USP2 O75604 1/20 0.58
TSHR P16473 1/20 0.58
HDAC3 O15379 1/20 0.57
HDAC4 P56524 1/20 0.57
HDAC1 Q13547 1/20 0.57
HDAC7 Q8WUI4 1/20 0.57
HDAC2 Q92769 1/20 0.57
HDAC10 Q969S8 1/20 0.57
HDAC11 Q96DB2 1/20 0.57
HDAC8 Q9BY41 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2007035 0.84 MEN1 (0.76) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL19002367 0.84 ALDH1A1 (0.76) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL9473705 0.82 LMNA (0.51) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL4780753 0.81 SMN1; SMN2 (0.72) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL14899353 0.81 ALDH1A1 (0.67) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL11003870 0.81 HTT (0.64) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL18997331 0.81 LMNA (0.69) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL11001127 0.80 KDM4E (0.53) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL1645833 0.80 ADRA2C (0.67) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL9191016 0.80 ALDH1A1 (0.65) ALDH1A1MEN1KMT2APOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4665239-B2 2011-04-06 JP claimed
EP-1417177-A4 ACYLSEMICARBAZIDES AS CYCLIN DEPENDENT KINASE INHIBITORS USEFUL AS ANTI-CANCER AND ANTI-PROLIFERATIVE AGENTS BRISTOL MYERS SQUIBB PHARMA CO (US) 2005-10-19 EP disclosed
EP-1417177-A2 ACYLSEMICARBAZIDES AS CYCLIN DEPENDENT KINASE INHIBITORS USEFUL AS ANTI-CANCER AND ANTI-PROLIFERATIVE AGENTS Bristol-Myers Squibb Pharma Company (US) 2004-05-12 EP disclosed
WO-2003007883-A2 ACYLSEMICARBAZIDES AS CYCLIN DEPENDENT KINASE INHIBITORS USEFUL AS ANTI-CANCER AND ANTI-PROLIFERATIVE AGENTS BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2003-01-30 WO disclosed
EP-1071668-A1 5-AMINOINDENO(1,2-C)PYRAZOL-4-ONES AS ANTI-CANCER AND ANTI-PROLIFERATIVE AGENTS Du Pont Pharmaceuticals Company (US) 2001-01-31 EP disclosed
WO-1999054308-A1 5-AMINOINDENO(1,2-C)PYRAZOL-4-ONES AS ANTI-CANCER AND ANTI-PROLIFERATIVE AGENTS DU PONT PHARMACEUTICALS COMPANY (US) 1999-10-28 WO disclosed