SCHEMBL16449166

SCHEMBL16449166

C=CCNC[C@@H](C)NS(=O)(=O)c1ccccc1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 2/20 0.43
SLC1A3 P43003 1/20 0.42
SLC1A2 P43004 1/20 0.42
SLC1A1 P43005 1/20 0.42
CASP1 P29466 3/20 0.39
ITGA2 P17301 1/20 0.38
NR3C1 P04150 1/20 0.38
ALDH1A1 P00352 6/20 0.38
TSHR P16473 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRK1 P41145 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL566412 0.81 CA1 (0.47) ALDH1A1LMNAHTTKMT2ASMN1; SMN2
SCHEMBL566411 0.81 CA1 (0.47) ALDH1A1LMNAHTTKMT2ASMN1; SMN2
SCHEMBL4070788 0.76 TSHR (0.49) ITGAVSLC1A3SLC1A2SLC1A1CASP1
SCHEMBL8851519 0.75 SLC1A3 (0.49) ITGAVSLC1A3SLC1A2SLC1A1CASP1
SCHEMBL9001208 0.72 SLC1A3 (0.55) ITGAVSLC1A3SLC1A2SLC1A1ITGA2
SCHEMBL8851832 0.71 SLC1A3 (0.54) ITGAVSLC1A3SLC1A2SLC1A1CASP1
SCHEMBL3865695 0.70 ALDH1A1 (0.35) ITGAVCASP1ALDH1A1TSHRLMNA
SCHEMBL20478178 0.70 SLC1A3 (0.53) ITGAVSLC1A3SLC1A2SLC1A1CASP1
SCHEMBL15352816 0.68 PKM (0.49) ITGAVSLC1A3SLC1A2SLC1A1ALDH1A1
SCHEMBL16825009 0.68 PKM (0.51) ITGAVSLC1A3SLC1A2SLC1A1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8951997-B2 Substituted isoquinoline derivative D. WESTERN THERAPEUTICS INSTITUTE, INC. (JP) 2015-02-10 US disclosed