SCHEMBL16456342

SCHEMBL16456342

Cc1ccc(-c2cnc(N)c(-c3ncc(F)cn3)c2)cc1

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 4/20 0.58
LRRK2 Q5S007 8/20 0.56
FYN P06241 3/20 0.51
TNKS O95271 1/20 0.49
TNKS2 Q9H2K2 1/20 0.49
USP7 Q93009 2/20 0.47
CHEK2 O96017 2/20 0.45
MKNK1 Q9BUB5 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16456297 0.84 MAP4K4 (0.61) MAP4K4LRRK2FYNTNKSTNKS2
SCHEMBL16456301 0.84 MAP4K4 (0.48) MAP4K4LRRK2FYNTNKSTNKS2
SCHEMBL4580922 0.79 MAP4K4 (0.54) MAP4K4LRRK2FYNUSP7CHEK2
SCHEMBL18393322 0.75 MAP4K4 (0.65) MAP4K4LRRK2FYNUSP7CHEK2
SCHEMBL11996767 0.74 ACHE (0.46)
SCHEMBL2967597 0.73 LRRK2 (0.55) MAP4K4LRRK2FYNUSP7
SCHEMBL28883695 0.73 MAP4K4 (0.61) MAP4K4LRRK2FYNUSP7
SCHEMBL29981431 0.73 MAP4K4 (0.61) MAP4K4LRRK2FYNUSP7
SCHEMBL16455993 0.72 CA12 (0.39) MAP4K4LRRK2FYNTNKSTNKS2
SCHEMBL13310774 0.71 MAP4K4 (0.39) MAP4K4LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9340549-B2 Oxazolidinone compounds and derivatives thereof AMGEN INC. (US) 2016-05-17 US disclosed
US-20150045368-A1 OXAZOLIDINONE COMPOUNDS AND DERIVATIVES THEREOF AMGEN INC. 2015-02-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150045368-A1 OXAZOLIDINONE COMPOUNDS AND DERIVATIVES THEREOF TNKS1BP1, TNKS, TBKBP1 MAP4K4 560/4885LRRK2 2305/4885FYN 404/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.