SCHEMBL16456392

SCHEMBL16456392

CCc1ccc(-c2cc(-c3ncccn3)c[nH]c2=O)cc1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TNKS O95271 7/20 0.49
TNKS2 Q9H2K2 1/20 0.49
ITK Q08881 2/20 0.44
PDGFRB P09619 1/20 0.42
ADRB2 P07550 1/20 0.38
DAO P14920 1/20 0.38
SLC6A7 Q99884 1/20 0.36
PDE2A O00408 1/20 0.35
NOTUM Q6P988 1/20 0.35
TTK P33981 1/20 0.35
AURKB Q96GD4 1/20 0.35
INCENP Q9NQS7 1/20 0.35
CTSV O60911 1/20 0.35
CTSL P07711 1/20 0.35
PARP1 P09874 1/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16456315 0.84 TNKS (0.52) TNKSTNKS2ITK
SCHEMBL16455971 0.81 TNKS (0.49) TNKSTNKS2ITK
SCHEMBL16456321 0.80 AURKA (0.56) TNKSITKPDGFRBDAOTTK
SCHEMBL16456338 0.79 TNKS (0.52) TNKSTNKS2ITKPDGFRBDAO
SCHEMBL10162103 0.75 ADRB2 (0.63) ADRB2SLC6A7TP53
SCHEMBL6535713 0.71 PARP1 (0.49) PDGFRBDAOTTKAURKBINCENP
SCHEMBL6692469 0.69 TNKS (0.44) TNKSTNKS2TTKAURKBINCENP
SCHEMBL16456296 0.69 TNKS (0.55) TNKSTNKS2TP53
SCHEMBL16456343 0.69 TNKS (0.41) TNKSPDGFRBDAONOTUMAURKB
SCHEMBL16456370 0.68 TNKS (0.53) TNKSTNKS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9340549-B2 Oxazolidinone compounds and derivatives thereof AMGEN INC. (US) 2016-05-17 US disclosed
US-20150045368-A1 OXAZOLIDINONE COMPOUNDS AND DERIVATIVES THEREOF AMGEN INC. 2015-02-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150045368-A1 OXAZOLIDINONE COMPOUNDS AND DERIVATIVES THEREOF TNKS1BP1, TNKS, TBKBP1 TNKS 2/4885TNKS2 10/4885ITK 350/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.