SCHEMBL6692469

SCHEMBL6692469

O=c1[nH]cc(-c2ncccn2)cc1-c1ccccc1-c1cccnc1F

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TNKS O95271 10/20 0.44
TNKS2 Q9H2K2 1/20 0.44
AURKA O14965 2/20 0.36
TTK P33981 2/20 0.36
AURKB Q96GD4 2/20 0.36
INCENP Q9NQS7 2/20 0.36
DHODH Q02127 1/20 0.35
CYP11B2 P19099 1/20 0.35
MAPT P10636 2/20 0.34
PTPRC P08575 1/20 0.34
METAP2 P50579 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6695727 0.78 MCL1 (0.47) TNKSTNKS2
SCHEMBL6692474 0.73 PARP1 (0.39) DHODHMAPTMETAP2
SCHEMBL16456315 0.72 TNKS (0.52) TNKSTNKS2MAPT
SCHEMBL16456392 0.69 TNKS (0.49) TNKSTNKS2TTKAURKBINCENP
SCHEMBL16455971 0.69 TNKS (0.49) TNKSTNKS2
SCHEMBL1887764 0.69 GRIA1 (0.52) TNKSDHODHMETAP2
SCHEMBL13314211 0.69 ALDH1A1 (0.49) MAPT
Hydrochloric Acid SCHEMBL3566887 0.68 ALDH1A1 (0.47) MAPT
SCHEMBL16160810 0.67 ALDH1A1 (0.41) TNKSTNKS2AURKATTKAURKB
SCHEMBL16151424 0.67 PKM (0.48) TNKSTNKS2AURKATTKAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465626-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING DIHYDROPYRIDINONE COMPOUNDS AND AN IMMUNOREGULATORY OR AN ANTIINFLAMMATORY AGENT AND THEIR USES Eisai Co., Ltd. (JP) 2004-10-13 EP disclosed
WO-2003047577-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING DIHYDROPYRIDINONE COMPOUNDS AND AN IMMUNOREGULATORY OR AN ANTIINFLAMMATORY AGENT AND THEIR USES EISAI CO LTD (JP) 2003-06-12 WO disclosed