SCHEMBL16456499

SCHEMBL16456499

CCc1ccc(S(=O)(=O)CCC(C)N(C)C2CCC(N)CC2)cc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40
CA2 P00918 1/20 0.37
RORC P51449 6/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
IL17A Q16552 2/20 0.33
PSIP1 O75475 1/20 0.33
CCR2 P41597 1/20 0.33
PTGDR Q13258 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
MMP1 P03956 1/20 0.33
MMP13 P45452 1/20 0.33
HSD11B1 P28845 1/20 0.33
MCHR1 Q99705 1/20 0.33
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2996925 1.00 HTR2A (0.40) HTR2AHTR2CCA2RORCMEN1
SCHEMBL16456530 0.87 POLB (0.38) MEN1KMT2ACCR2MMP1MMP13
SCHEMBL2992306 0.87 POLB (0.38) MEN1KMT2ACCR2MMP1MMP13
SCHEMBL2991411 0.86 KMT2A (0.37) HTR2AHTR2CMEN1KMT2APSIP1
SCHEMBL5753723 0.86 KMT2A (0.37) HTR2AHTR2CMEN1KMT2APSIP1
SCHEMBL16456497 0.71 CCR2 (0.49) HTR2AHTR2CCCR2
SCHEMBL2996923 0.71 CCR2 (0.49) HTR2AHTR2CCCR2
SCHEMBL29296587 0.71 CA2 (0.50) CA2MEN1KMT2APSIP1MMP1
SCHEMBL22254882 0.70 SLC6A4 (0.33) HTR2AHTR2CMCHR1
SCHEMBL5033532 0.66 OPRM1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1620391-B1 CYCLIC DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL MYERS SQUIBB CO (US) 2014-01-15 EP disclosed