SCHEMBL1645805

SCHEMBL1645805

O=C(O)c1ccccc1-c1c2ccc(=O)c(Cl)c-2oc2c(Cl)c(O)ccc12

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GNG2 P59768 4/20 0.70
GNB1 P62873 4/20 0.70
PTPN7 P35236 1/20 0.58
FTO Q9C0B1 2/20 0.46
USP2 O75604 2/20 0.46
KDM4A O75164 1/20 0.46
NSD2 O96028 1/20 0.46
ALPL P05186 1/20 0.46
PLCG1 P19174 1/20 0.46
TNNI3 P19429 1/20 0.46
NFKB1 P19838 1/20 0.46
TNNT2 P45379 1/20 0.46
MMP14 P50281 1/20 0.46
CASP6 P55212 1/20 0.46
TNNC1 P63316 1/20 0.46
KDM4C Q9H3R0 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
SOS1 Q07889 2/20 0.43
MEN1 O00255 2/20 0.43
THRB P10828 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10293755 0.85 GNG2 (0.56) GNG2GNB1PTPN7FTOUSP2
SCHEMBL2777300 0.82 GNG2 (1.00) GNG2GNB1PTPN7FTOUSP2
SCHEMBL15424239 0.80 GNG2 (0.70) GNG2GNB1PTPN7FTOUSP2
SCHEMBL14001247 0.80 GNG2 (0.70) GNG2GNB1PTPN7FTOUSP2
SCHEMBL29588006 0.80 GNG2 (0.70) GNG2GNB1PTPN7FTOUSP2
SCHEMBL6125804 0.80 GNG2 (0.70) GNG2GNB1PTPN7FTOUSP2
SCHEMBL21611728 0.79 GNG2 (0.69) GNG2GNB1PTPN7FTOUSP2
SCHEMBL14030799 0.78 GNG2 (0.67) GNG2GNB1PTPN7FTOUSP2
SCHEMBL840931 0.77 KDM4A (0.44) GNG2GNB1PTPN7USP2KDM4A
SCHEMBL8948052 0.76 GNG2 (0.65) GNG2GNB1PTPN7FTOUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 97 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240315965-A1 COMPOSITIONS AND METHODS RELATED TO PHARMACEUTICAL EXCIPIENTS Natural Extraction Systems, LLC (US) 2024-09-26 US claimed
WO-2022182527-A1 COMPOSITIONS AND METHODS RELATED TO PHARMACEUTICAL EXCIPIENTS Natural Extraction Systems, LLC (US) 2022-09-01 WO claimed
EP-1192450-B1 HIGH ENERGY PHOTOTHERAPEUTIC AGENTS PROVECTUS PHARMATECH INC (US) 2014-12-03 EP claimed
EP-1753467-B1 DIAGNOSTIC AGENTS FOR POSITRON EMISSION IMAGING USING RADIOLABELED HALOGENATED XANTHENES AND METHODS FOR POSITRON EMISSION IMAGING WITH RADIOLABELED HALOGENATED XANTHENE DIAGNOSTIC AGENTS PROVECTUS PHARMATECH INC (US) 2013-01-09 EP claimed
US-7427389-B2 Diagnostic agents for positron emission imaging using radiolabeled halogenated xanthenes PROVECTUS PHARMATECH, INC. (US) 2008-09-23 US claimed
EP-1753467-A4 DIAGNOSTIC AGENTS FOR POSITRON EMISSION IMAGING USING RADIOLABELED HALOGENATED XANTHENES AND METHODS FOR POSITRON EMISSION IMAGING WITH RADIOLABELED HALOGENATED XANTHENE DIAGNOSTIC AGENTS XANTECH PHARMACEUTICALS INC (US) 2008-09-17 EP claimed
EP-1311261-B1 MEDICAMENTS FOR CHEMOTHERAPEUTIC TREATMENT OF DISEASE PHOTOGEN INC (US) 2008-01-23 EP claimed
EP-1753467-A1 DIAGNOSTIC AGENTS FOR POSITRON EMISSION IMAGING USING RADIOLABELED HALOGENATED XANTHENES AND METHODS FOR POSITRON EMISSION IMAGING WITH RADIOLABELED HALOGENATED XANTHENE DIAGNOSTIC AGENTS Xantech Pharmaceuticals, Inc. (US) 2007-02-21 EP claimed
WO-2006001925-A1 DIAGNOSTIC AGENTS FOR POSITRON EMISSION IMAGING USING RADIOLABELED HALOGENATED XANTHENES AND METHODS FOR POSITRON EMISSION IMAGING WITH RADIOLABELED HALOGENATED XANTHENE DIAGNOSTIC AGENTS XANTECH PHARMACEUTICALS, INC. (US) 2006-01-05 WO claimed
US-20050276752-A1 Diagnostic agents for positron emission imaging using radiolabeled halogenated xanthenes XANTECH PHARMACEUTICALS, INC. 2005-12-15 US claimed
EP-1292298-A1 INTRACORPOREAL MEDICAMENTS FOR HIGH ENERGY PHOTOTHERAPEUTIC TREATMENT OF DISEASE Photogen, Inc. (US) 2003-03-19 EP claimed
EP-1284727-A1 INTRACORPOREAL MEDICAMENTS FOR PHOTODYNAMIC TREATMENT OF DISEASE Photogen, Inc. (US) 2003-02-26 EP claimed
US-20020161035-A1 Medicaments for chemotherapeutic treatment of disease PHOTOGEN, INC. 2002-10-31 US claimed
EP-1210078-A1 IMPROVED TOPICAL MEDICAMENTS AND METHODS FOR PHOTODYNAMIC TREATMENT OF DISEASE Photogen, Inc. (US) 2002-06-05 EP claimed
WO-2002005812-A1 MEDICAMENTS FOR CHEMOTHERAPEUTIC TREATMENT OF DISEASE PHOTOGEN, INC. (US) 2002-01-24 WO claimed
US-20020001567-A1 Intracorporeal medicaments for high energy phototherapeutic treatment of disease PHOTOGEN, INC. 2002-01-03 US claimed
WO-2001076595-A1 INTRACORPOREAL MEDICAMENTS FOR HIGH ENERGY PHOTOTHERAPEUTIC TREATMENT OF DISEASE PHOTOGEN, INC. (US) 2001-10-18 WO claimed
WO-2001072301-A1 INTRACORPOREAL MEDICAMENTS FOR PHOTODYNAMIC TREATMENT OF DISEASE PHOTOGEN, INC. (US) 2001-10-04 WO claimed
US-20010022970-A1 Intracorporeal medicaments for photodynamic treatment of disease PHOTOGEN, INC. 2001-09-20 US claimed
WO-2001012181-A1 IMPROVED TOPICAL MEDICAMENTS AND METHODS FOR PHOTODYNAMIC TREATMENT OF DISEASE PHOTOGEN, INC. (US) 2001-02-22 WO claimed