SCHEMBL1645813

SCHEMBL1645813

COc1ccccc1N(CCO)C(=O)CN

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LIMK1 P53667 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.42
PABPC1 P11940 1/20 0.42
HTT P42858 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
TSHR P16473 1/20 0.40
POLB P06746 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ACHE P22303 1/20 0.40
CTSD P07339 1/20 0.40
SNCA P37840 1/20 0.39
TSPO P30536 1/20 0.39
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29138562 0.83 ADORA2A (0.45) LIMK1SMN1; SMN2HTTALDH1A1POLB
SCHEMBL9133783 0.82 TDP1 (0.44) SMN1; SMN2L3MBTL1ALDH1A1KDM4EPOLB
SCHEMBL11267655 0.81 ALDH1A1 (0.47) SMN1; SMN2PABPC1HTTL3MBTL1ALDH1A1
SCHEMBL9135231 0.78 POLB (0.43) SMN1; SMN2L3MBTL1ALDH1A1KDM4EPOLB
SCHEMBL30994803 0.78 ADORA2A (0.47) SMN1; SMN2PABPC1HTTALDH1A1TSPO
SCHEMBL9134080 0.77 ALDH1A1 (0.47) L3MBTL1ALDH1A1POLBTSPO
SCHEMBL11266461 0.76 ALDH1A1 (0.45) SMN1; SMN2PABPC1L3MBTL1ALDH1A1KDM4E
SCHEMBL11258983 0.76 ALDH1A1 (0.45) SMN1; SMN2PABPC1L3MBTL1ALDH1A1KDM4E
SCHEMBL5965849 0.74 AOC3 (0.45) SMN1; SMN2ALDH1A1TSHRCTSDLMNA
SCHEMBL8710643 0.74 LMNA (0.63) SMN1; SMN2HTTL3MBTL1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4665239-B2 2011-04-06 JP claimed
EP-1417177-A4 ACYLSEMICARBAZIDES AS CYCLIN DEPENDENT KINASE INHIBITORS USEFUL AS ANTI-CANCER AND ANTI-PROLIFERATIVE AGENTS BRISTOL MYERS SQUIBB PHARMA CO (US) 2005-10-19 EP disclosed
EP-1417177-A2 ACYLSEMICARBAZIDES AS CYCLIN DEPENDENT KINASE INHIBITORS USEFUL AS ANTI-CANCER AND ANTI-PROLIFERATIVE AGENTS Bristol-Myers Squibb Pharma Company (US) 2004-05-12 EP disclosed
WO-2003007883-A2 ACYLSEMICARBAZIDES AS CYCLIN DEPENDENT KINASE INHIBITORS USEFUL AS ANTI-CANCER AND ANTI-PROLIFERATIVE AGENTS BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2003-01-30 WO disclosed
EP-1071668-A1 5-AMINOINDENO(1,2-C)PYRAZOL-4-ONES AS ANTI-CANCER AND ANTI-PROLIFERATIVE AGENTS Du Pont Pharmaceuticals Company (US) 2001-01-31 EP disclosed
WO-1999054308-A1 5-AMINOINDENO(1,2-C)PYRAZOL-4-ONES AS ANTI-CANCER AND ANTI-PROLIFERATIVE AGENTS DU PONT PHARMACEUTICALS COMPANY (US) 1999-10-28 WO disclosed