SCHEMBL8710643

SCHEMBL8710643

COc1cccc(C(=O)N(CCO)c2ccccc2OC)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.63
HTT P42858 2/20 0.53
GAA P10253 1/20 0.49
HPGD P15428 1/20 0.49
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
MAPK1 P28482 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.46
PARP1 P09874 1/20 0.46
THRB P10828 2/20 0.45
ALDH1A1 P00352 2/20 0.45
TSPO P30536 1/20 0.45
KDM4E B2RXH2 1/20 0.45
HSD17B10 Q99714 1/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
TP53 P04637 1/20 0.45
CDK4 P11802 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8713891 0.85 LMNA (0.64) LMNAHTTGAAHPGDCES2
SCHEMBL6784816 0.80 PTGES (0.60) LMNAHTTMAPK1SMN1; SMN2ALDH1A1
SCHEMBL8713421 0.78 LMNA (0.53) LMNAHTTHPGDMAPK1SMN1; SMN2
SCHEMBL29138562 0.78 ADORA2A (0.45) LMNAHTTSMN1; SMN2ALDH1A1TSPO
SCHEMBL9230549 0.76 HSD11B1 (0.57) LMNAHTTSMN1; SMN2ALDH1A1KMT2A
SCHEMBL15835211 0.75 KDM4E (0.50) LMNAHTTGAAHPGDMAPK1
SCHEMBL1645813 0.74 LIMK1 (0.44) LMNAHTTL3MBTL1SMN1; SMN2ALDH1A1
SCHEMBL1926940 0.74 TRPM8 (0.53) LMNAHPGDCES2CES1MAPK1
SCHEMBL6778747 0.73 NPC1 (0.55) LMNAMAPK1TDP1SMN1; SMN2ALDH1A1
SCHEMBL21425705 0.72 MEN1 (0.60) HPGDCES2CES1MAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed