SCHEMBL16463000

SCHEMBL16463000

Cn1ccc2ccc(-n3ccc(=O)c4ccccc43)cc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BIRC5 O15392 1/20 0.42
CYP2A6 P11509 1/20 0.41
PER2 O15055 1/20 0.40
CRY1 Q16526 1/20 0.40
CRY2 Q49AN0 1/20 0.40
HPGD P15428 1/20 0.39
LPAR5 Q9H1C0 1/20 0.39
CFTR P13569 1/20 0.38
CA12 O43570 1/20 0.38
BRD4 O60885 1/20 0.38
BRPF1 P55201 1/20 0.38
CA9 Q16790 1/20 0.38
KAT2B Q92831 1/20 0.38
BRD9 Q9H8M2 1/20 0.38
PTPN1 P18031 1/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
MAOB P27338 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30462932 0.81 ALDH1A1 (0.46) BIRC5HPGDALDH1A1GAA
SCHEMBL16463633 0.79 HTR6 (0.47) BRD4KDM4E
SCHEMBL29576413 0.77 ALDH1A1 (0.59) HPGDPTPN1KDM4EALDH1A1MAPT
SCHEMBL1809581 0.77 ALDH1A1 (0.59) HPGDPTPN1KDM4EALDH1A1MAPT
Iodide SCHEMBL27839552 0.75 ALDH1A1 (0.57) HPGDPTPN1KDM4EALDH1A1MAPT
Hydrochloric Acid SCHEMBL29744398 0.75 ALDH1A1 (0.57) HPGDPTPN1KDM4EALDH1A1MAPT
SCHEMBL26684188 0.74 CRBN (0.53) CYP2A6LPAR5CFTRMAPTPRKCI
SCHEMBL7662776 0.73 COMT (0.49) BIRC5HPGDKDM4E
SCHEMBL16464432 0.73 MAPT (0.41) HPGDKDM4EALDH1A1MAPTNQO2
SCHEMBL16464557 0.73 KDM4E (0.40) BIRC5HPGDKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8629162-B2 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-01-14 US disclosed