SCHEMBL1646835

SCHEMBL1646835

NC(=O)c1cc(-c2cn(C3CCCCO3)nc2-c2cccc(Cl)c2)ccn1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BRAF P15056 1/20 0.38
CNR2 P34972 5/20 0.38
NUDT1 P36639 2/20 0.38
ABL1 P00519 1/20 0.36
USP30 Q70CQ3 1/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
BTK Q06187 1/20 0.35
GRM5 P41594 1/20 0.35
ATR Q13535 1/20 0.34
EGFR P00533 1/20 0.34
FYN P06241 1/20 0.34
GRM2 Q14416 1/20 0.34
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1647453 0.90 CNR2 (0.41) BRAFCNR2NUDT1ABL1NPC1
SCHEMBL1645154 0.88 EGFR (0.41) BRAFCNR2ATREGFR
SCHEMBL1646821 0.85 MAPK14 (0.41) BRAFABL1BTKATREGFR
SCHEMBL1645150 0.84 CSNK1D (0.40) BRAFABL1BTKATR
SCHEMBL1646703 0.77 NUDT1 (0.53) BRAFNUDT1TP53
SCHEMBL26112994 0.76 TP53 (0.38) ABL1NPC1RAB9AGRM5TP53
SCHEMBL1646072 0.75 MCL1 (0.42) BRAFABL1
SCHEMBL1649098 0.74 ABL1 (0.41) BRAFABL1
SCHEMBL22075459 0.72 FGFR3 (0.37) BRAFABL1GRM5ATRTP53
SCHEMBL1646854 0.72 FGFR1 (0.42) BRAFABL1ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2784070-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784073-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784071-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784072-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2308866-A1 Phenylpyri(mi)dinylpyrazoles and their use as fungicides Bayer CropScience AG (DE) 2011-04-13 EP disclosed